SCHEMBL7730638

SCHEMBL7730638

Cc1ccc(Cl)c(OC2CCN(C(=O)[C@@H]3CC(NC(=O)CNC(=O)OC(C)(C)C)CN3C(=O)OC(C)(C)C)CC2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 1/20 0.41
MCHR1 Q99705 1/20 0.41
CYP1A2 P05177 1/20 0.38
POLB P06746 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
LMNA P02545 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TGM2 P21980 1/20 0.36
EPHX2 P34913 1/20 0.36
GPR6 P46095 1/20 0.36
TOP2A P11388 1/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
PDE4B Q07343 4/20 0.35
ALDH1A1 P00352 2/20 0.35
PDE4A P27815 2/20 0.35
PDE4C Q08493 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7730647 1.00 NPBWR1 (0.41) NPBWR1MCHR1CYP1A2POLBCYP3A4
SCHEMBL7730651 1.00 NPBWR1 (0.41) NPBWR1MCHR1CYP1A2POLBCYP3A4
SCHEMBL7722091 0.86 STS (0.37) NPBWR1MCHR1TGM2CTSLCTSB
SCHEMBL7722100 0.86 STS (0.37) NPBWR1MCHR1TGM2CTSLCTSB
SCHEMBL7722247 0.86 STS (0.37) NPBWR1MCHR1TGM2CTSLCTSB
SCHEMBL7722098 0.86 STS (0.37) NPBWR1MCHR1TGM2CTSLCTSB
SCHEMBL7722007 0.80 TGM2 (0.42) LMNATGM2MEN1KMT2A
SCHEMBL7722009 0.80 TGM2 (0.42) LMNATGM2MEN1KMT2A
SCHEMBL7722003 0.80 TGM2 (0.42) LMNATGM2MEN1KMT2A
SCHEMBL7730983 0.79 MCL1 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399629-B1 PYRROLIDINES AND PIPERIDINES FOR TREATING MICROBIAL INFECTIONS BY REDUCING EXPORT OF COADMINISTERED ANTIMICROBIAL AGENT OR COMPOUND SYNTHESIZED BY MICROBES FOR THEIR GROWTH; REDUCING IN VIVO AVAILABILITY MICROCIDE PHARMACEUTICALS, INC. 2002-06-04 US disclosed