SCHEMBL7732264

SCHEMBL7732264

CC(=O)c1ccc(-c2ccc(C#Cc3ccccc3)cc2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.70
SMN1; SMN2 Q16637 1/20 0.70
HSD17B1 P14061 1/20 0.53
LMNA P02545 2/20 0.53
GRM5 P41594 2/20 0.49
HPGD P15428 2/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP1A1 P04798 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP1B1 Q16678 1/20 0.48
ACACB O00763 2/20 0.48
MMP2 P08253 1/20 0.47
MMP9 P14780 1/20 0.47
MMP12 P39900 1/20 0.47
MMP14 P50281 1/20 0.47
MMP15 P51511 1/20 0.47
MMP16 P51512 1/20 0.47
MMP26 Q9NRE1 1/20 0.47
VCP P55072 1/20 0.47
FFAR1 O14842 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL400497 0.94 MAPT (0.59) MAPTSMN1; SMN2LMNAGRM5HPGD
SCHEMBL7252924 0.83 MAPT (1.00) MAPTSMN1; SMN2HSD17B1LMNAHPGD
SCHEMBL7738989 0.83 MAPT (1.00) MAPTSMN1; SMN2HSD17B1LMNAHPGD
SCHEMBL51207 0.83 MAPT (1.00) MAPTSMN1; SMN2HSD17B1LMNAHPGD
SCHEMBL15960257 0.82 RARB (0.63) MAPTSMN1; SMN2LMNAHPGDALDH1A1
SCHEMBL28933332 0.81 HPGD (0.50) MAPTSMN1; SMN2LMNAGRM5HPGD
Water SCHEMBL9631565 0.81 MAPT (0.95) MAPTSMN1; SMN2HSD17B1LMNAHPGD
Hydrogen Sulfide SCHEMBL28388826 0.81 MAPT (0.95) MAPTSMN1; SMN2HSD17B1LMNAHPGD
Acetophenone SCHEMBL27985201 0.81 MAPT (0.86) MAPTSMN1; SMN2HSD17B1LMNAHPGD
SCHEMBL12445832 0.80 MAPT (0.59) MAPTSMN1; SMN2LMNAALDH1A1CYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7790744-B2 Cyclic peptide antifungal agents and process for preparation thereof ELI LILLY AND COMPANY (US) 2010-09-07 US disclosed
US-6743777-B1 TRISPHENYL ACYL DERIVATIVES OF THE ECHINOCANDIN CLASS; CANDIDA ALBICANS; ANTIFUNGAL AND ANTIPARASITIC; CYCLIC HEXAPEPTIDES HAVING UNIQUE SIDE CHAIN ACYL GROUP ELI LILLY AND COMPANY 2004-06-01 US disclosed