SCHEMBL7732335

SCHEMBL7732335

N[C@H](CCc1ccccc1)c1nc(C(=O)O)co1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.49
ANPEP P15144 2/20 0.41
ERAP1 Q9NZ08 2/20 0.41
ERAP2 Q6P179 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
DAGLA Q9Y4D2 4/20 0.39
FAAH O00519 1/20 0.39
PTPN1 P18031 1/20 0.39
KMT2A Q03164 1/20 0.37
METAP2 P50579 1/20 0.37
METAP1 P53582 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6466167 0.85 CES1 (0.46) CES1ANPEPERAP1ERAP2HDAC1
SCHEMBL7732052 0.79 RAB9A (0.43) HDAC1HDAC8HDAC6KMT2AMETAP2
SCHEMBL7732103 0.76 RAB9A (0.53) HDAC1HDAC8HDAC6KMT2A
SCHEMBL7735836 0.76 SLC1A3 (0.40) KMT2AMETAP2
SCHEMBL6463614 0.76 HDAC1 (0.45) CES1HDAC1HDAC8HDAC6FAAH
SCHEMBL5168702 0.75 HDAC1 (0.43) CES1HDAC1HDAC8HDAC6PTPN1
SCHEMBL7723269 0.73 MAPT (0.48) KMT2A
SCHEMBL6463446 0.73 DAGLA (0.51) CES1ERAP2HDAC1HDAC8HDAC6
SCHEMBL25387512 0.71 HDAC1 (0.40) CES1HDAC1HDAC8HDAC6PTPN1
SCHEMBL2078861 0.70 HDAC1 (0.54) CES1HDAC1HDAC8HDAC6PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436980-B1 TRANSPORT PROTEIN SUPPRESSORS; MICROBIOCIDES ESSENTIAL THERAPEUTICS, INC. 2002-08-20 US disclosed
US-6204279-B1 SECONDARY AMIDE CONTAINING BENZOXAZOLE DERIVATIVES MICROCIDE PHARMACEUTICALS, INC. 2001-03-20 US disclosed