SCHEMBL7733429

SCHEMBL7733429

Nc1cnc2ccc(Cc3ccccc3)cc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
MAPT P10636 2/20 0.42
GAA P10253 1/20 0.42
PKM P14618 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
KLKB1 P03952 3/20 0.42
MAP4K1 Q92918 3/20 0.42
TLR9 Q9NR96 1/20 0.40
LTA4H P09960 1/20 0.40
IDH1 O75874 1/20 0.40
AOC3 Q16853 1/20 0.39
CALM1 P0DP23 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
TSHR P16473 1/20 0.39
CASP1 P29466 1/20 0.39
HTT P42858 1/20 0.39
ATM Q13315 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL8136028 0.88 KLKB1 (0.42) KLKB1MAP4K1
SCHEMBL22926854 0.87 PDE10A (0.49) KDM4EMAPTGAAPKMTDP1
SCHEMBL20524060 0.78 EGFR (0.41) KDM4EMAPTGAAKLKB1MAP4K1
SCHEMBL7727062 0.78 SMN1; SMN2 (0.48) KDM4EMAPTGAAKLKB1MAP4K1
SCHEMBL7728250 0.77 MGAM (0.62) IDH1
SCHEMBL27824234 0.75 MET (0.53) KDM4EMAPTALDH1A1TP53HSP90AA1
SCHEMBL30503636 0.74 EGFR (0.61) KDM4EMAPTGAATDP1TLR9
SCHEMBL11162210 0.74 EGFR (0.61) KDM4EMAPTGAATDP1TLR9
SCHEMBL23330368 0.74 KDM4E (0.40) KDM4EMAPTGAAKLKB1MAP4K1
SCHEMBL5799847 0.74 NOS1 (0.41) KDM4EMAPTKLKB1MAP4K1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399629-B1 PYRROLIDINES AND PIPERIDINES FOR TREATING MICROBIAL INFECTIONS BY REDUCING EXPORT OF COADMINISTERED ANTIMICROBIAL AGENT OR COMPOUND SYNTHESIZED BY MICROBES FOR THEIR GROWTH; REDUCING IN VIVO AVAILABILITY MICROCIDE PHARMACEUTICALS, INC. 2002-06-04 US disclosed
WO-2000001714-A1 EFFLUX PUMP INHIBITORS MICROCIDE PHARMACEUTICALS, INC. (US) 2000-01-13 WO disclosed