SCHEMBL7733803

SCHEMBL7733803

N[C@H](CCc1ccccc1)C(O)c1nc2cc(CC3CC3)ccc2s1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.35
NPC1 O15118 1/20 0.35
NFKB1 P19838 1/20 0.35
STAT1 P42224 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
METAP2 P50579 5/20 0.34
METAP1 P53582 3/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
HIF1A Q16665 1/20 0.34
HSD17B10 Q99714 1/20 0.34
KDM4E B2RXH2 1/20 0.34
LIPC P11150 2/20 0.34
LIPG Q9Y5X9 3/20 0.33
S1PR1 P21453 2/20 0.33
S1PR3 Q99500 2/20 0.33
LOXL2 Q9Y4K0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7735956 0.86 S1PR1 (0.39) HPGDNPC1NFKB1STAT1RAB9A
SCHEMBL7731411 0.81 HPGD (0.51) HPGDNPC1NFKB1RAB9ANFKB2
SCHEMBL7735562 0.72 S1PR1 (0.39) HPGDNPC1NFKB1STAT1RAB9A
Hydrochloric Acid SCHEMBL7347434 0.67 HPGD (0.52) HPGDNPC1NFKB1RAB9ANFKB2
Hydrochloric Acid SCHEMBL6356550 0.67 HPGD (0.52) HPGDNPC1NFKB1RAB9ANFKB2
SCHEMBL7730593 0.66 AAK1 (0.49) HPGDNPC1NFKB1STAT1RAB9A
SCHEMBL6632792 0.66 LOXL2 (0.56) HPGDNPC1NFKB1RAB9ANFKB2
SCHEMBL7735961 0.65 LOXL2 (0.51) HPGDNPC1NFKB1RAB9ANFKB2
SCHEMBL7733999 0.64 IDO1 (0.43) HPGDNPC1RAB9AMETAP2METAP1
SCHEMBL6651863 0.64 LOXL2 (0.60) HPGDNPC1RAB9ACYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436980-B1 TRANSPORT PROTEIN SUPPRESSORS; MICROBIOCIDES ESSENTIAL THERAPEUTICS, INC. 2002-08-20 US disclosed
US-6204279-B1 SECONDARY AMIDE CONTAINING BENZOXAZOLE DERIVATIVES MICROCIDE PHARMACEUTICALS, INC. 2001-03-20 US disclosed