SCHEMBL773469

SCHEMBL773469

FC(F)(F)C(Br)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
TRPA1 O75762 1/20 0.41
DPP4 P27487 2/20 0.38
TSHR P16473 2/20 0.38
ALDH1A1 P00352 2/20 0.38
F2 P00734 1/20 0.38
HSD17B10 Q99714 1/20 0.36
HTR2A P28223 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
ACP3 P15309 1/20 0.34
CYP2D6 P10635 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7394160 1.00 CES2 (0.41) CES2CES1TRPA1DPP4TSHR
SCHEMBL8728321 0.78 ALDH1A1 (0.33) CES2CES1TRPA1TSHRALDH1A1
SCHEMBL10590024 0.78 CES2 (0.44) CES2CES1TRPA1DPP4TSHR
SCHEMBL28477107 0.77 CYP2A6 (0.40) DPP4ALDH1A1HSD17B10HTR2ACYP2D6
SCHEMBL14321447 0.77 IDO1 (0.39) ALDH1A1HSD17B10
SCHEMBL14321076 0.75 CHRNA7 (0.39) TSHRALDH1A1HSD17B10MEN1KMT2A
SCHEMBL5866912 0.75 GSK3B (0.35) ALDH1A1HSD17B10
SCHEMBL14321453 0.75 TSHR (0.44) TSHRALDH1A1HSD17B10
SCHEMBL29488208 0.75 HDAC4 (0.42) CES2CES1
SCHEMBL14321085 0.75 HDAC4 (0.42) CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 450 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119264013-A Preparation method of (1-arylmethyl-3-aryl-1-trifluoromethyl propyl) aromatic compound 南京工业大学 2025-01-07 CN claimed
CN-118344340-A Quinolinone compound containing 1,2, 4-triazole or 1,3, 4-oxadiazole structure and preparation and application thereof 贵州大学 2024-07-16 CN claimed
CN-117486852-A Fluorine-containing rotaxane molecule and preparation method and application thereof 中国科学院精密测量科学与技术创新研究院 2024-02-02 CN claimed
CN-114806260-B Preparation method of modified nano zinc oxide filler, hydrophobic antifouling coating and preparation method thereof 海南大学 2023-02-28 CN claimed
CN-114988981-A Preparation method of alpha-trifluoromethyl arylpropyne compound 盐城工学院 2022-09-02 CN claimed
CN-113549062-B Chiral quaternary ammonium salt phase transfer catalyst with high steric hindrance derived from cinchona alkaloid and synthesis method thereof 南京工业大学 2022-08-09 CN claimed
CN-114806260-A Preparation method of modified nano zinc oxide filler, hydrophobic antifouling coating and preparation method thereof 海南大学 2022-07-29 CN claimed
CN-108395396-B Preparation method of chiral o-amino alcohol intermediate, antagonist and analogue thereof 复旦大学 2021-07-23 CN claimed
CN-109438461-B Tuliquiritigenin A derivative with anti-leukemia activity and preparation method and application thereof 广西中医药大学 2021-04-20 CN claimed
CN-104987338-A Low cost method for preparing sitagliptin phosphate salt key intermediate XINFA PHARMACEUTICAL CO LTD 2015-10-21 CN claimed
US-8901365-B2 Catalytic Wittig and Mitsunobu reactions BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2014-12-02 US claimed
CN-100569746-C Arylbis (perfluoroalkylsulfonyl) methane and metal salts thereof, and process for producing the same JAPAN SCIENCE & TECH AGENCY (JP) 2009-12-16 CN claimed
CN-1481357-A Arylbis (perfluoroalkylsulfonyl) methane and metal salts thereof, and process for producing the same 科学技术振兴事业团 2004-03-10 CN claimed
WO-2025120200-A1 NEW ANTI-INFECTIVE TRICYCLIC SPIROLACTAMS COMPOUNDS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 2025-06-12 WO disclosed
CN-119264013-A Preparation method of (1-arylmethyl-3-aryl-1-trifluoromethyl propyl) aromatic compound 南京工业大学 2025-01-07 CN disclosed
WO-2024230104-A1 POLYCYCLIC COMPOUND AND USE THEREOF 浙江同源康医药股份有限公司 2024-11-14 WO disclosed
US-5248689-A Hypotensive agents, congestive heart failure, renal failure or glaucoma SMITHKLINE BEECHAM CORPORATION (US) 1993-09-28 US disclosed
WO-1993001160-A1 AROMATIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY MERCK SHARP & DOHME LIMITED (GB) 1993-01-21 WO disclosed
US-4966987-A CHEMICAL INTERMEDIATE FOR FLUORINATED AROMATIC COMPOUND HOECHST AKTIENGESELLSCHAFT (DE) 1990-10-30 US disclosed
US-4132737-A ENZYME INHIBITORS ELI LILLY AND COMPANY (US) 1979-01-02 US disclosed