SCHEMBL7735112

SCHEMBL7735112

CS(=O)(=O)c1ccc(-c2nn(Cc3cccnc3)c(=S)cc2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.54
PTGS1 P23219 9/20 0.54
MARS1 P56192 2/20 0.44
JAK2 O60674 2/20 0.44
PTK2 Q05397 2/20 0.44
SLC16A3 O15427 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3948221 0.89 PTGS2 (0.57) PTGS2PTGS1MARS1JAK2PTK2
SCHEMBL395735 0.84 MARS1 (0.43) PTGS2PTGS1MARS1SLC16A3
SCHEMBL3946879 0.81 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL3938737 0.79 MEN1 (0.57) PTGS2PTGS1
SCHEMBL396392 0.79 MEN1 (0.43)
SCHEMBL3939882 0.77 MARS1 (0.46) PTGS2PTGS1MARS1SLC16A3
SCHEMBL5577174 0.76 MARS1 (0.45) PTGS2PTGS1MARS1SLC16A3
SCHEMBL393900 0.74 MARS1 (0.47) PTGS2PTGS1MARS1SLC16A3
SCHEMBL3945552 0.73 MEN1 (0.44) MARS1SLC16A3
SCHEMBL3940435 0.73 PTGS2 (0.61) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6348468-B1 THESE COMPOUNDS HAVE EXCELLENT INHIBITORY ACTIVITY AGAINST INTERLEUKIN-1.BETA. PRODUCTION, IMMUNE SYSTEM DISEASES, INFLAMMATORY DISEASES, ISCHEMIC DISEASES AND THE LIKE. KOWA CO., LTD. (JP) 2002-02-19 US claimed