SCHEMBL7737816

SCHEMBL7737816

CC(C)(C)C(=O)Nc1nc2c(c(=O)[nH]1)CC(CCc1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s1)CN2

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GART P22102 12/20 0.57
DHFR P00374 1/20 0.52
ATIC P31939 3/20 0.47
FOLR1 P15328 8/20 0.46
SLC46A1 Q96NT5 5/20 0.46
FOLR2 P14207 3/20 0.46
SLC19A1 P41440 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7745908 0.87 GART (0.75) GARTATICFOLR1SLC46A1FOLR2
SCHEMBL9382790 0.86 DHFR (0.52) GARTDHFRATICFOLR1SLC46A1
SCHEMBL9382796 0.86 DHFR (0.52) GARTDHFRATICFOLR1SLC46A1
SCHEMBL6900553 0.80 GART (0.47) GARTDHFRATICFOLR1
SCHEMBL9380609 0.80 DHFR (0.59) GARTDHFRATICFOLR1SLC46A1
SCHEMBL9381796 0.80 DHFR (0.59) GARTDHFRATICFOLR1SLC46A1
SCHEMBL9383067 0.80 DHFR (0.59) GARTDHFRATICFOLR1SLC46A1
SCHEMBL1065440 0.80 GART (0.62) GARTATICFOLR1SLC46A1FOLR2
SCHEMBL20659947 0.80 GART (0.62) GARTATICFOLR1SLC46A1FOLR2
SCHEMBL14403392 0.80 DHFR (0.59) GARTDHFRATICFOLR1SLC46A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6426417-B1 CYCLIZATION OF A CYANO-ESTER DERIVATIVE WITH 2,6-DIAMINO-6-HYDROXYPYRIMIDINE IN THE PRESENCE OF ACETIC ACID AND ACETONITRILE ELI LILLY AND COMPANY 2002-07-30 US disclosed