SCHEMBL7738443

SCHEMBL7738443

C=CCc1cc(C[C@](C)(NC(C)=O)C(=O)O)c2ccccc2c1[SiH](C)C

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.33
ALDH1A1 P00352 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD17B10 Q99714 2/20 0.32
MMP2 P08253 1/20 0.31
MMP13 P45452 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7738413 0.75 PPARA (0.36) ALDH1A1CYP3A4CYP2C9CYP2C19HSD17B10
SCHEMBL7736596 0.71 MEN1 (0.33) ALDH1A1HSD17B10KDM4EMEN1KMT2A
SCHEMBL2331138 0.66 ALDH1A1 (0.53) ALDH1A1CYP3A4CYP2C9CYP2C19HSD17B10
SCHEMBL2329888 0.66 ALDH1A1 (0.53) ALDH1A1CYP3A4CYP2C9CYP2C19HSD17B10
SCHEMBL8410894 0.66 ALDH1A1 (0.53) ALDH1A1CYP3A4CYP2C9CYP2C19HSD17B10
SCHEMBL3485811 0.61 NAALAD2 (0.41) ALDH1A1CYP3A4CYP2C9CYP2C19MEN1
SCHEMBL28268750 0.60 MEN1 (0.39) ELANEALDH1A1CYP2C9HSD17B10KDM4E
SCHEMBL17911429 0.59 CYP3A4 (0.72) ALDH1A1CYP3A4CYP2C9CYP2C19HSD17B10
SCHEMBL27914028 0.59 CYP3A4 (0.72) ALDH1A1CYP3A4CYP2C9CYP2C19HSD17B10
SCHEMBL22033119 0.59 BLM (0.56) ALDH1A1CYP3A4HSD17B10KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6416861-B1 COMBINATORIAL CHEMISTRY NORTHWESTERN UNIVERSITY 2002-07-09 US disclosed
WO-2000049022-A2 ORGANOSILICON COMPOUNDS AND USES THEREOF NORTHWESTERN UNIVERSITY (US) 2000-08-24 WO disclosed