SCHEMBL7738848

SCHEMBL7738848

O=C(O)c1nc2cc(Cl)ccc2cc1O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.46
PIM2 Q9P1W9 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
KMO O15229 1/20 0.45
DYRK1A Q13627 1/20 0.43
ALDH1A1 P00352 5/20 0.42
KDM4E B2RXH2 2/20 0.42
IGFBP3 P17936 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
MAPT P10636 1/20 0.41
DAO P14920 1/20 0.40
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
CASP1 P29466 1/20 0.39
PTGES O14684 1/20 0.39
ALOX5 P09917 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
CASP7 P55210 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17913386 0.85 ALDH1A1 (0.46) PIM1PIM2CA1CA2KMO
SCHEMBL6565660 0.85 KMT2A (0.43) PIM1PIM2CA1CA2KMO
SCHEMBL8802100 0.84 DYRK1A (0.47) PIM1PIM2CA1CA2KMO
SCHEMBL30556744 0.84 DYRK1A (0.47) PIM1PIM2CA1CA2KMO
SCHEMBL8574083 0.83 ALDH1A1 (0.47) PIM1PIM2CA1CA2KMO
SCHEMBL4658383 0.82 KMO (0.39) PIM1PIM2CA1CA2KMO
SCHEMBL29093592 0.81 KMO (0.53) PIM1PIM2KMODYRK1AALDH1A1
SCHEMBL705432 0.79 EGLN1 (0.56)
SCHEMBL3988553 0.79 PIM1 (0.37) PIM1PIM2CA1CA2KMO
SCHEMBL31028951 0.79 EGLN1 (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329497-B1 ANTITUMOR AGENTS; VIRICIDES AGAINST HUMAN IMMUNODEFICIENCY VIRUS THE SCRIPPS RESEARCH INSTITUTE 2001-12-11 US disclosed
EP-0996458-A4 SANDRAMYCIN ANALOGS SCRIPPS RESEARCH INST (US) 2001-05-02 EP disclosed
EP-0996458-A1 SANDRAMYCIN ANALOGS The Scripps Research Institute (US) 2000-05-03 EP disclosed
WO-1998043663-A1 SANDRAMYCIN ANALOGS THE SCRIPPS RESEARCH INSTITUTE (US) 1998-10-08 WO disclosed
CN-1062905-A 4-hydroxyl-7-chloro-quinolinic acid synthetic method TANG LIANGPING (CN) 1992-07-22 CN disclosed