SCHEMBL7739646

SCHEMBL7739646

Cc1c([N+](=O)[O-])cc(Br)c(F)c1CNC(=O)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
LMNA P02545 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ALDH1A1 P00352 3/20 0.36
GLA P06280 1/20 0.36
HPGD P15428 1/20 0.36
ALOX12 P18054 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP1A2 P05177 1/20 0.35
AR P10275 3/20 0.34
PGR P06401 1/20 0.32
CYP3A4 P08684 1/20 0.32
MAPT P10636 2/20 0.31
THRB P10828 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
GSTO1 P78417 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7740445 0.82 MEN1 (0.39) MEN1KMT2ALMNAL3MBTL1ALDH1A1
SCHEMBL7880767 0.81 HPGD (0.36) MEN1KMT2ALMNAL3MBTL1ALDH1A1
SCHEMBL25834987 0.76 AR (0.36) MEN1KMT2ALMNAL3MBTL1ALDH1A1
SCHEMBL27564256 0.75 MEN1 (0.36) MEN1KMT2ALMNAL3MBTL1ALDH1A1
SCHEMBL7880691 0.71 AR (0.41) MEN1KMT2ALMNAL3MBTL1ALDH1A1
SCHEMBL29570831 0.70 L3MBTL1 (0.45) MEN1KMT2ALMNAL3MBTL1ALDH1A1
SCHEMBL13277233 0.70 L3MBTL1 (0.45) MEN1KMT2ALMNAL3MBTL1ALDH1A1
SCHEMBL9677433 0.69 CYP1A2 (0.48) ALDH1A1SMN1; SMN2CYP1A2CYP3A4MAPT
SCHEMBL13277488 0.69 CYP1A2 (0.41) MEN1KMT2ALMNAL3MBTL1ALDH1A1
SCHEMBL31381636 0.69 CYP1A2 (0.41) MEN1KMT2ALMNAL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1217928-C Heterocyclic compound having NOS inhibitory action CHUGAI SEIYAKA K K (JP) 2005-09-07 CN disclosed
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
CN-1280565-A Heterocyclic compounds having NOS inhibitory activities CHUGAI SEIYAKA K K (JP) 2001-01-17 CN disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed