SCHEMBL7740445

SCHEMBL7740445

Cc1c([N+](=O)[O-])cc(Br)c(F)c1CNC(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
EPAS1 Q99814 1/20 0.36
AAK1 Q2M2I8 2/20 0.35
CA12 O43570 3/20 0.35
CA1 P00915 3/20 0.35
CA2 P00918 3/20 0.35
CA9 Q16790 3/20 0.35
KDM4A O75164 1/20 0.35
ALDH1A1 P00352 1/20 0.34
ADRA2A P08913 1/20 0.34
DRD5 P21918 1/20 0.34
DRD3 P35462 1/20 0.34
P2RY6 Q15077 1/20 0.34
BCHE P06276 1/20 0.34
CNR2 P34972 1/20 0.34
CYP1A2 P05177 1/20 0.33
RPS6KA1 Q15418 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7880092 0.83 EPAS1 (0.40) MEN1LMNAKMT2AL3MBTL1EPAS1
SCHEMBL7739646 0.82 MEN1 (0.41) MEN1LMNAKMT2AL3MBTL1ALDH1A1
SCHEMBL7740423 0.78 ALDH1A1 (0.37) MEN1LMNAKMT2AL3MBTL1CA12
SCHEMBL27564256 0.74 MEN1 (0.36) MEN1LMNAKMT2AL3MBTL1ALDH1A1
SCHEMBL7872397 0.74 EPAS1 (0.35) MEN1LMNAKMT2AEPAS1CA12
SCHEMBL31716307 0.72 EPAS1 (0.45) LMNAL3MBTL1EPAS1AAK1CA12
SCHEMBL19717777 0.71 POLB (0.49) LMNAKDM4AALDH1A1CYP1A2MAPT
SCHEMBL18300499 0.71 AAK1 (0.44) LMNAL3MBTL1EPAS1AAK1CA12
SCHEMBL30868193 0.70 PDGFRB (0.46) MEN1LMNAKMT2ACA12CA1
SCHEMBL28355220 0.70 AAK1 (0.41) MEN1LMNAKMT2AL3MBTL1AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1217928-C Heterocyclic compound having NOS inhibitory action CHUGAI SEIYAKA K K (JP) 2005-09-07 CN disclosed
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
CN-1280565-A Heterocyclic compounds having NOS inhibitory activities CHUGAI SEIYAKA K K (JP) 2001-01-17 CN disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed