SCHEMBL7740698

SCHEMBL7740698

CC(=O)O[C@@H]1[C@H](OC(C)=O)[C@@H](C)O[C@H]1n1c(NC(C)C)nc2cc(F)c(F)cc21

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.41
ACACB O00763 3/20 0.35
ADORA2B P29275 4/20 0.33
MT-CO1 P00395 2/20 0.33
MT-CO2 P00403 2/20 0.33
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
EDNRA P25101 1/20 0.32
OPRM1 P35372 1/20 0.32
HTR2B P41595 1/20 0.32
KCNH2 Q12809 1/20 0.32
IDH1 O75874 4/20 0.31
MCHR1 Q99705 1/20 0.30
CA9 Q16790 2/20 0.30
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7742267 0.92 HDAC6 (0.47) HDAC6ACACBKCNH2
SCHEMBL7734423 0.92 HDAC6 (0.47) HDAC6ACACBIDH1
SCHEMBL7114252 0.88 HDAC6 (0.34) HDAC6ACACB
SCHEMBL7118668 0.86 ACACB (0.36) HDAC6ACACB
SCHEMBL7215084 0.86 LMNA (0.46) HDAC6CA9CA12CA1CA2
SCHEMBL7215090 0.86 LMNA (0.46) HDAC6CA9CA12CA1CA2
SCHEMBL7121805 0.84 HDAC6 (0.45) HDAC6MCHR1
SCHEMBL7115119 0.84 HDAC6 (0.46) HDAC6
SCHEMBL7117894 0.83 HDAC6 (0.48) HDAC6
SCHEMBL7117899 0.83 HDAC6 (0.41) HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6413938-B1 HERPES VIRUS THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2002-07-02 US disclosed
EP-0970100-A1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 2000-01-12 EP disclosed
WO-1998035977-A1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 1998-08-20 WO disclosed