SCHEMBL7742065

SCHEMBL7742065

CCOC(=O)[C@H](Cc1ccc(NS(C)(=O)=O)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTPRB P23467 9/20 0.49
HPGD P15428 1/20 0.48
RECQL P46063 1/20 0.48
CTSS P25774 6/20 0.46
CTSK P43235 5/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HTT P42858 1/20 0.46
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
CTSL P07711 1/20 0.45
CTSB P07858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31689469 0.91 KLK5 (0.52) PTPRBCTSSCTSKCTSLCTSB
SCHEMBL7736843 0.88 PTPRB (0.47) PTPRBCTSSCTSKCYP1A2CYP2C9
SCHEMBL3820732 0.87 ACE (0.57) PTPRBCTSSCTSKCTSLCTSB
SCHEMBL7988834 0.86 BCL2 (0.55) PTPRBCTSSCTSKALDH1A1CTSL
SCHEMBL25095271 0.86 LMNA (0.57) PTPRBRECQLALDH1A1
SCHEMBL14803767 0.84 PPARG (0.53) HPGDCTSSCTSKCYP1A2CYP2C9
SCHEMBL20045974 0.84 PPARG (0.53) HPGDCTSSCTSKCYP1A2CYP2C9
SCHEMBL1826124 0.84 ITGB3 (0.48) CTSSCTSKCYP1A2CYP2C9CYP2C19
SCHEMBL1826126 0.84 ITGB3 (0.48) CTSSCTSKCYP1A2CYP2C9CYP2C19
SCHEMBL7742078 0.84 HDAC8 (0.48) CTSSCTSKCYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023025861-A1 NEW VASHS INHIBITORS, CONJUGATES THEREOF AND THEIR USES AS DRUGS OR AS RESEARCH TOOLS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2023-03-02 WO disclosed
US-6420424-B1 ADMINISTERING PHENYLALANINE AMIDE DERIVATIVES (SUCH AS S-ETHYL-2-AMINO-3-(4-CHLOROPHENYL)PROPIONATE HYDROCHLORIDE) TO TREAT ALLERGIC DISORDERS, INCLUDING ASTHMA, RHINITIS, DERMATITUS, AND PRURITIS SMITHKLINE BEECHAM CORPORATION 2002-07-16 US disclosed