SCHEMBL7742519

SCHEMBL7742519

NC(=O)NC1C=Cc2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.36
HTR6 P50406 1/20 0.36
LMNA P02545 2/20 0.34
TSHR P16473 2/20 0.34
MAPK1 P28482 2/20 0.34
SCN4A P35499 1/20 0.34
SCN5A Q14524 1/20 0.34
SCN9A Q15858 1/20 0.34
ATM Q13315 2/20 0.33
NR3C1 P04150 1/20 0.32
KMT2A Q03164 2/20 0.32
CYP2D6 P10635 1/20 0.32
MEN1 O00255 1/20 0.32
CYP2C9 P11712 2/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
GFER P55789 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3601520 0.84 HTR2A (0.33) HTR2AHTR6LMNAATMKMT2A
SCHEMBL3601522 0.84 MEN1 (0.36) HTR2AHTR6LMNAATMKMT2A
SCHEMBL835707 0.82 MTNR1A (0.39) HTR2ALMNAATMKMT2ACYP2D6
SCHEMBL4510570 0.82 HTR2A (0.36) HTR2AHTR6LMNATSHRKMT2A
SCHEMBL28106726 0.81 HTR6 (0.32) HTR2AHTR6LMNAATMKMT2A
SCHEMBL11593035 0.79 IDO1 (0.38) LMNATSHRKMT2AMEN1MAPT
SCHEMBL1920068 0.78 SSTR1 (0.36) LMNANR3C1KMT2AMEN1NPSR1
SCHEMBL4510567 0.75 HTR6 (0.33) HTR2AHTR6LMNACYP2D6SIGMAR1
SCHEMBL28244022 0.75 HTR2A (0.42) HTR2AHTR6LMNAKMT2ACYP2D6
SCHEMBL6542107 0.74 HTR2A (0.40) HTR2AHTR6LMNAKMT2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2002512230-A 2002-04-23 JP claimed
EP-1071668-A1 5-AMINOINDENO(1,2-C)PYRAZOL-4-ONES AS ANTI-CANCER AND ANTI-PROLIFERATIVE AGENTS Du Pont Pharmaceuticals Company (US) 2001-01-31 EP claimed
WO-1999054308-A1 5-AMINOINDENO(1,2-C)PYRAZOL-4-ONES AS ANTI-CANCER AND ANTI-PROLIFERATIVE AGENTS DU PONT PHARMACEUTICALS COMPANY (US) 1999-10-28 WO claimed