SCHEMBL7743329

SCHEMBL7743329

CC(N)c1ccccc1-c1cccc(O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 1/20 0.46
MIF P14174 1/20 0.46
HTR2A P28223 1/20 0.46
ADRA1A P35348 1/20 0.46
HTR2B P41595 1/20 0.46
HSD17B1 P14061 7/20 0.44
HSD17B2 P37059 7/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
ADRA2A P08913 3/20 0.41
ADRA2B P18089 3/20 0.41
ADRA2C P18825 3/20 0.41
PLK4 O00444 1/20 0.41
ROCK2 O75116 1/20 0.41
RPS6KA5 O75582 1/20 0.41
MAP4K4 O95819 1/20 0.41
RET P07949 1/20 0.41
PDGFRB P09619 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7743489 0.98 ADRB1 (0.45) ADRB1MIFHTR2AADRA1AHTR2B
SCHEMBL10094321 0.86 HSD17B1 (0.47) HTR2BHSD17B1HSD17B2CYP3A4CYP2C9
SCHEMBL11133836 0.81 AKR1C3 (0.47) HSD17B1HSD17B2CYP3A4CYP2C9AKR1C3
SCHEMBL26307961 0.79 CA12 (0.46) CYP3A4ADRA2AADRA2C
SCHEMBL1254511 0.79 CA12 (0.46) CYP3A4ADRA2AADRA2C
SCHEMBL28472426 0.79 AKR1C3 (0.58) CYP2C9AKR1C3AKR1C2ADRA2BBAZ2B
SCHEMBL11479928 0.79 HSD17B1 (0.40) HSD17B1HSD17B2CYP3A4CYP2C9AKR1C3
SCHEMBL4745768 0.77 AKR1C3 (0.41) AKR1C3AKR1C2ADRA2AADRA2BADRA2C
SCHEMBL4779452 0.77 HSD17B1 (0.64) HSD17B1HSD17B2CYP3A4CYP2C9PLK4
Boric Acid SCHEMBL28704756 0.77 CA12 (0.41) CYP3A4ADRA2AADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091736-A4 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO INC (US) 2001-10-24 EP disclosed
EP-1091736-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2001-04-18 EP disclosed
WO-2000001382-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2000-01-13 WO disclosed