Isoniazid

Isoniazid

SCHEMBL7744265

NC(N)=O.NNC(=O)c1ccncc1

nearest known ligand 0.91

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

inhA

The experimentally established mechanism targets of Isoniazid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.91
CYP3A4 P08684 3/20 0.91
MPO P05164 2/20 0.91
CYP1A2 P05177 2/20 0.91
CYP2D6 P10635 2/20 0.91
CYP2C19 P33261 2/20 0.91
ADORA3 P0DMS8 1/20 0.91
CYP2A6 P11509 1/20 0.91
ALDH1A1 P00352 4/20 0.61
CA1 P00915 1/20 0.58
CA9 Q16790 1/20 0.58
MAPT P10636 3/20 0.55
TDP1 Q9NUW8 1/20 0.55
GAA P10253 1/20 0.55
HIF1A Q16665 2/20 0.54
KDM5A P29375 1/20 0.54
BLM P54132 1/20 0.54
GFER P55789 1/20 0.54
PMP22 Q01453 1/20 0.54
L3MBTL1 Q9Y468 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isoniazid SCHEMBL2390873 0.96 KDM4E (1.00) KDM4ECYP3A4MPOCYP1A2CYP2D6
Isoniazid SCHEMBL12264078 0.96 KDM4E (1.00) KDM4ECYP3A4MPOCYP1A2CYP2D6
Isoniazid SCHEMBL2072618 0.96 KDM4E (1.00) KDM4ECYP3A4MPOCYP1A2CYP2D6
Isoniazid SCHEMBL228 0.96 KDM4E (1.00) KDM4ECYP3A4MPOCYP1A2CYP2D6
Isoniazid SCHEMBL16642161 0.96 KDM4E (1.00) KDM4ECYP3A4MPOCYP1A2CYP2D6
Isoniazid SCHEMBL16642160 0.96 KDM4E (1.00) KDM4ECYP3A4MPOCYP1A2CYP2D6
Isoniazid SCHEMBL12264083 0.96 KDM4E (1.00) KDM4ECYP3A4MPOCYP1A2CYP2D6
Isoniazid SCHEMBL12264081 0.96 KDM4E (1.00) KDM4ECYP3A4MPOCYP1A2CYP2D6
Isoniazid SCHEMBL7502798 0.93 KDM4E (0.95) KDM4ECYP3A4MPOCYP1A2CYP2D6
Isoniazid SCHEMBL20958129 0.93 KDM4E (0.95) KDM4ECYP3A4MPOCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1017999-A4 PROCESSES FOR PREPARING BARRIER LAYER FILMS FOR USE IN ENZYME ELECTRODES AND FILMS MADE THEREBY YSI INC (US) 2001-09-26 EP disclosed
EP-1017999-A1 PROCESSES FOR PREPARING BARRIER LAYER FILMS FOR USE IN ENZYME ELECTRODES AND FILMS MADE THEREBY YSI INCORPORATED (US) 2000-07-12 EP disclosed
WO-1997035185-A1 PROCESSES FOR PREPARING BARRIER LAYER FILMS FOR USE IN ENZYME ELECTRODES AND FILMS MADE THEREBY YSI INCORPORATED (US) 1997-09-25 WO disclosed