SCHEMBL7744958

SCHEMBL7744958

Cc1ccc(Cn2nc(C)cc2C(=O)O)cc1.NC(=O)c1ccc(Cl)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.61
NPSR1 Q6W5P4 1/20 0.61
P2RY14 Q15391 4/20 0.53
RAB9A P51151 4/20 0.51
NPC1 O15118 3/20 0.51
KMT2A Q03164 2/20 0.51
POLB P06746 1/20 0.50
NAMPT P43490 1/20 0.49
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC10 Q969S8 1/20 0.48
HDAC11 Q96DB2 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
HDAC9 Q9UKV0 1/20 0.48
HDAC5 Q9UQL6 1/20 0.48
NCOR2 Q9Y618 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
4-Chloroaniline SCHEMBL7744962 0.88 MAPT (0.64) MAPTNPSR1P2RY14RAB9ANPC1
SCHEMBL6258641 0.88 MAPT (0.64) MAPTNPSR1P2RY14RAB9ANPC1
SCHEMBL2079137 0.86 MAPT (0.62) MAPTNPSR1P2RY14RAB9ANPC1
SCHEMBL7744333 0.80 GRN (0.76) MAPTNPSR1NPC1GRNSORT1
SCHEMBL5178107 0.77 GRN (0.67) MAPTNPSR1RAB9ANPC1KMT2A
SCHEMBL7744959 0.76 NPSR1 (1.00) MAPTNPSR1P2RY14RAB9ANPC1
SCHEMBL22000813 0.76 HDAC3 (0.55) MAPTNPSR1P2RY14RAB9ANPC1
SCHEMBL10150650 0.74 MAPT (0.53) MAPTNPSR1RAB9ANPC1KMT2A
SCHEMBL12585876 0.73 PTGER4 (0.64) MAPTNPSR1
SCHEMBL18435242 0.73 PTGER4 (0.64) MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1252156-A1 BLOCKADE OF VOLTAGE DEPENDENT SODIUM CHANNELS University College London (GB) 2002-10-30 EP disclosed
WO-2001057024-A1 BLOCKADE OF VOLTAGE DEPENDENT SODIUM CHANNELS UNIVERSITY COLLEGE LONDON (GB) 2001-08-09 WO disclosed