SCHEMBL7746303

SCHEMBL7746303

CC(=O)[C@@H]1CCCN1c1nc(-c2ccccc2)nc2[nH]ccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.46
ADORA3 P0DMS8 1/20 0.46
ADORA2A P29274 1/20 0.46
ADORA2B P29275 1/20 0.46
PIK3CA P42336 3/20 0.42
MTOR P42345 3/20 0.42
KMT2A Q03164 2/20 0.41
JAK3 P52333 2/20 0.41
ELANE P08246 2/20 0.39
TSHR P16473 2/20 0.39
ALDH1A1 P00352 2/20 0.39
USP2 O75604 1/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C9 P11712 1/20 0.39
ALOX15 P16050 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4083747 0.89 ELANE (0.51) ADORA1ADORA3ADORA2AADORA2BPIK3CA
SCHEMBL7752203 0.82 ADORA1 (0.47) ADORA1ADORA3ADORA2AADORA2BPIK3CA
SCHEMBL4084126 0.77 MAT2A (0.47) KMT2AELANETSHRALDH1A1USP2
SCHEMBL4078297 0.77 MAT2A (0.47) KMT2AELANETSHRALDH1A1USP2
SCHEMBL7751006 0.76 MAT2A (0.46) KMT2AELANETSHRNUDT1TP53
SCHEMBL5189246 0.74 ADORA1 (0.47) ADORA1ADORA3ADORA2AADORA2BPIK3CA
SCHEMBL8355465 0.74 ADORA1 (0.47) ADORA1ADORA3ADORA2AADORA2BPIK3CA
SCHEMBL2825572 0.74 ADORA1 (0.47) ADORA1ADORA3ADORA2AADORA2BPIK3CA
SCHEMBL4077312 0.74 ADORA1 (0.47) ADORA1ADORA3ADORA2AADORA2BPIK3CA
SCHEMBL7749780 0.73 MAT2A (0.47) KMT2AELANETSHRNUDT1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6680324-B2 4-AMINO-6-PHENYL-PYRROLO(2,3-D)PYRIMIDINE DERIVATIVES OSI PHARMACEUTICALS, INC. 2004-01-20 US disclosed