SCHEMBL7747406

SCHEMBL7747406

CC(C)(C)OC(=O)N1CCC(N2CCC3(CC2)OC(=O)Nc2ccc(Cl)cc23)CC1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.44
F11 P03951 10/20 0.44
AVPR1A P37288 1/20 0.42
ELOVL6 Q9H5J4 1/20 0.40
STS P08842 2/20 0.40
CNR1 P21554 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
CALCRL Q16602 1/20 0.39
MAPK8 P45983 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4760270 0.91 F11 (0.50) F11AVPR1A
SCHEMBL3276637 0.87 CALCRL (0.46) HRH3AVPR1AMAPTCALCRL
SCHEMBL17205370 0.85 F11 (0.55) F11AVPR1A
SCHEMBL18490941 0.81 F11 (0.53) F11
SCHEMBL17205822 0.81 F11 (0.53) F11
SCHEMBL5003859 0.79 PLD2 (0.44) F11AVPR1AKDM4EMAPTTHRB
SCHEMBL2103144 0.76 AVPR1A (0.50) AVPR1AMAPTCALCRL
SCHEMBL13314901 0.76 CALCRL (0.50) F11AVPR1AKDM4EMAPTCALCRL
SCHEMBL10914505 0.76 AVPR1A (0.50) F11AVPR1AELOVL6
SCHEMBL13314907 0.74 KCNH2 (0.56) AVPR1AKDM4ECALCRL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001022919-A2 SPIRO[BICYCLIC -AZACYCLOALKYL AND -CYCLOALKYL] DERIVATIVES AND USES THEREOF MERCK & CO., INC. (US) 2001-04-05 WO disclosed