SCHEMBL7748729

SCHEMBL7748729

CN(C)CCCCc1ccccn1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 2/20 0.58
SIGMAR1 Q99720 1/20 0.52
KDM4E B2RXH2 2/20 0.50
TSHR P16473 2/20 0.50
TDP1 Q9NUW8 2/20 0.50
NPSR1 Q6W5P4 1/20 0.50
HRH3 Q9Y5N1 1/20 0.50
POLB P06746 1/20 0.50
NAAA Q02083 1/20 0.49
CYP2C19 P33261 4/20 0.49
CYP2D6 P10635 2/20 0.49
LMNA P02545 1/20 0.49
TAAR1 Q96RJ0 1/20 0.49
ALDH1A1 P00352 1/20 0.49
ALOX15 P16050 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.48
MAPT P10636 1/20 0.48
LIN28A Q9H9Z2 1/20 0.48
CHRM2 P08172 1/20 0.47
CHRM4 P08173 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18042405 0.98 HRH1 (0.61) HRH1SIGMAR1KDM4ETSHRTDP1
SCHEMBL2681263 0.94 HRH1 (0.55) HRH1KDM4ETSHRTDP1NPSR1
SCHEMBL30086100 0.86 KDM4E (0.58) HRH1KDM4ETSHRTDP1NPSR1
SCHEMBL229256 0.86 KDM4E (0.58) HRH1KDM4ETSHRTDP1NPSR1
Hydrochloric Acid SCHEMBL29367467 0.85 KDM4E (0.57) HRH1KDM4ETSHRTDP1NPSR1
SCHEMBL726512 0.84 HRH1 (0.76) HRH1TDP1HRH3NAAACYP2C19
SCHEMBL23761760 0.83 HRH1 (0.51) HRH1KDM4ETSHRTDP1NPSR1
SCHEMBL4418086 0.82 HRH1 (0.80) HRH1TDP1HRH3NAAACYP2C19
SCHEMBL2843489 0.82 HRH1 (0.80) HRH1TDP1HRH3NAAACYP2C19
SCHEMBL31040594 0.82 HRH1 (0.80) HRH1TDP1HRH3NAAACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1069901-A4 CALCILYTIC COMPOUNDS AND METHOD OF USE SMITHKLINE BEECHAM CORP (US) 2001-06-13 EP disclosed
EP-1069901-A1 CALCILYTIC COMPOUNDS AND METHOD OF USE SMITHKLINE BEECHAM CORPORATION (US) 2001-01-24 EP disclosed
WO-1999051241-A1 CALCILYTIC COMPOUNDS AND METHOD OF USE SMITHKLINE BEECHAM CORPORATION (US) 1999-10-14 WO disclosed