SCHEMBL7749402

SCHEMBL7749402

C/C=C/C(=O)Nc1ccc(Br)cc1Br

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.50
TP53 P04637 1/20 0.50
MAPT P10636 1/20 0.50
POLB P06746 2/20 0.48
NPC1 O15118 2/20 0.47
HPGD P15428 1/20 0.47
NFKB1 P19838 1/20 0.47
RAB9A P51151 1/20 0.47
NFKB2 Q00653 1/20 0.47
RELA Q04206 1/20 0.47
ALDH1A1 P00352 2/20 0.45
GAA P10253 1/20 0.45
THRB P10828 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
EGFR P00533 4/20 0.43
TRPM2 O94759 1/20 0.43
PELI1 Q96FA3 1/20 0.43
ERBB2 P04626 2/20 0.42
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7749404 1.00 SMN1; SMN2 (0.50) SMN1; SMN2TP53MAPTPOLBNPC1
SCHEMBL22501856 0.87 MEN1 (0.48) SMN1; SMN2TP53MAPTPOLBALDH1A1
SCHEMBL22501857 0.87 MEN1 (0.48) SMN1; SMN2TP53MAPTPOLBALDH1A1
SCHEMBL28820634 0.79 EGFR (0.66) SMN1; SMN2TP53MAPTNPC1RAB9A
SCHEMBL31236185 0.77 ALDH1A1 (0.62) SMN1; SMN2MAPTPOLBNPC1HPGD
SCHEMBL1801329 0.77 ALDH1A1 (0.62) SMN1; SMN2MAPTPOLBNPC1HPGD
SCHEMBL31236186 0.77 ALDH1A1 (0.62) SMN1; SMN2MAPTPOLBNPC1HPGD
SCHEMBL30499697 0.73 KIF11 (0.51) SMN1; SMN2MAPTNPC1HPGDNFKB1
SCHEMBL9835752 0.73 NPC1 (0.53) SMN1; SMN2MAPTNPC1HPGDNFKB1
SCHEMBL6823604 0.73 KIF11 (0.51) SMN1; SMN2MAPTNPC1HPGDNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1071658-A2 BTK INHIBITORS AND METHODS FOR THEIR IDENTIFICATION AND USE Parker Hughes Institute (US) 2001-01-31 EP disclosed
WO-1999054286-A2 BTK INHIBITORS AND METHODS FOR THEIR IDENTIFICATION AND USE PARKER HUGHES INSTITUTE (US) 1999-10-28 WO disclosed