SCHEMBL7751410

SCHEMBL7751410

OC(CNc1ccccc1)CN1CCN(CCCCC(c2ccc(F)cc2)c2ccc(F)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 5/20 0.47
SLC6A4 P31645 3/20 0.47
DRD3 P35462 3/20 0.47
HTR2A P28223 2/20 0.47
ADRA1A P35348 2/20 0.47
HRH1 P35367 2/20 0.47
OPRD1 P41143 2/20 0.47
OPRK1 P41145 2/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2D6 P10635 2/20 0.47
DRD4 P21917 2/20 0.47
CACNA1F O60840 1/20 0.47
DRD1 P21728 1/20 0.47
DRD5 P21918 1/20 0.47
HRH2 P25021 1/20 0.47
ADRA1D P25100 1/20 0.47
HTR2C P28335 1/20 0.47
HTR7 P34969 1/20 0.47
ADRA1B P35368 1/20 0.47
OPRM1 P35372 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7543312 0.99 MEN1 (0.48) SLC6A3SLC6A4DRD3HTR2AADRA1A
SCHEMBL4760958 0.97 CYP3A4 (0.51) SLC6A3SLC6A4DRD3HTR2AADRA1A
SCHEMBL8615736 0.97 CYP3A4 (0.51) SLC6A3SLC6A4DRD3HTR2AADRA1A
SCHEMBL8616378 0.97 CYP3A4 (0.51) SLC6A3SLC6A4DRD3HTR2AADRA1A
Hydrochloric Acid SCHEMBL7543578 0.96 MEN1 (0.52) SLC6A3SLC6A4DRD3HTR2AADRA1A
Hydrochloric Acid SCHEMBL8867248 0.96 MEN1 (0.52) SLC6A3SLC6A4DRD3HTR2AADRA1A
SCHEMBL8677737 0.94 SCN5A (0.51) SLC6A3SLC6A4DRD3HTR2AADRA1A
SCHEMBL7754343 0.92 CYP3A4 (0.53) SLC6A3SLC6A4DRD3HTR2AADRA1A
SCHEMBL7755959 0.92 SLC6A3 (0.50) SLC6A3SLC6A4DRD3DRD4DRD2
Hydrochloric Acid SCHEMBL7543310 0.91 SLC6A3 (0.49) SLC6A3SLC6A4DRD3DRD4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0706796-B1 DOPAMINE RE-UPTAKE INHIBITORS FOR THE TREATMENT OF PARKINSON'S SYNDROME POLA CHEM IND INC (JP) 2001-02-28 EP claimed
US-5747493-A N-/DIPHENYLALKYL/-PIPERAZINYL-2-HYDROXYPROPYLAMINES POLA CHEMICAL INDUSTRIES, INC. (JP) 1998-05-05 US claimed
EP-0706796-A1 DOPAMINE REINCORPORATION INHIBITOR POLA CHEMICAL INDUSTRIES, INC. (JP) 1996-04-17 EP claimed