SCHEMBL7751683

SCHEMBL7751683

N=C(N)NCCC[C@@H](NC(=O)C(c1ccccc1)c1ccccc1)C(=O)NCc1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NPY1R P25929 18/20 0.62
NPY5R Q15761 3/20 0.62
NPY4R P50391 3/20 0.62
NPY2R P49146 1/20 0.62
NPFFR1 Q9GZQ6 2/20 0.61
NPFFR2 Q9Y5X5 2/20 0.61
MCHR1 Q99705 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6899864 0.95 NPY1R (0.71) NPY1RNPY5RNPY4RNPY2RNPFFR1
SCHEMBL7059807 0.95 NPY1R (0.71) NPY1RNPY5RNPY4RNPY2RNPFFR1
SCHEMBL7746012 0.94 NPY1R (0.61) NPY1RNPY5RNPY4RNPY2RNPFFR1
SCHEMBL4651828 0.94 NPY1R (0.61) NPY1RNPY5RNPY4RNPY2RNPFFR1
SCHEMBL650331 0.94 NPY1R (0.72) NPY1RNPY5RNPY4RNPFFR1NPFFR2
SCHEMBL4653108 0.93 NPY1R (0.60) NPY1RNPY5RNPY4RNPY2RNPFFR1
SCHEMBL4651993 0.93 NPY1R (0.68) NPY1RNPY5RNPY4RNPY2RNPFFR1
SCHEMBL7039837 0.93 NPY1R (0.60) NPY1RNPY5RNPY4RNPY2RNPFFR1
SCHEMBL4653159 0.93 NPY1R (0.60) NPY1RNPY5RNPY4RNPY2RNPFFR1
SCHEMBL8112679 0.93 NPY1R (0.58) NPY1RNPY5RNPY4RNPY2RNPFFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0680469-B1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME BOEHRINGER INGELHEIM PHARMA (DE) 2000-04-26 EP claimed
US-6313128-B1 CAN BE USED AS LYPOLYSIS/LYPOGENESIS REGULATORS IN THE SKIN WITHOUT, INTERFERRING WITH THE SKIN'S NATURAL FUNCTIONS; FOR THERAPY OF SABORRHEA AND ACNE SANOFI-SYNTHELABO (FR) 2001-11-06 US disclosed
EP-0680469-B1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME BOEHRINGER INGELHEIM PHARMA (DE) 2000-04-26 EP disclosed