SCHEMBL7752019

SCHEMBL7752019

O=C(O)C(CC1CCCCC1)c1ccc(OCc2ccc3ccccc3n2)cc1

nearest known ligand 0.71

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 20/20 0.71
HDAC6 Q9UBN7 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9556595 0.99 ALOX5 (0.71) ALOX5HDAC6
SCHEMBL7751568 0.95 ALOX5 (0.67) ALOX5HDAC6
SCHEMBL8799856 0.91 ALOX5 (0.65) ALOX5HDAC6
SCHEMBL9430813 0.89 ALOX5 (0.64) ALOX5HDAC6
SCHEMBL9556694 0.88 ALOX5 (0.63) ALOX5HDAC6
SCHEMBL9148914 0.88 ALOX5 (0.62) ALOX5HDAC6
Veliflapon SCHEMBL7752617 0.86 ALOX5 (0.71) ALOX5HDAC6
SCHEMBL9556500 0.84 ALOX5 (0.58) ALOX5HDAC6
SCHEMBL2109295 0.83 ALOX5 (1.00) ALOX5HDAC6
SCHEMBL7818344 0.83 ALOX5 (1.00) ALOX5HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5358955-A Antiinflammatory agents ABBOTT LABORATORIES (US) 1994-10-25 US claimed
WO-2001035960-A1 USE OF SUBSTITUTED 4-(QUINOLIN 2-YL-METHOXY)PHENYL-ACETIC ACID DERIVATIVES FOR THE TREATMENT OF DISEASES BAYER AKTIENGESELLSCHAFT (DE) 2001-05-25 WO disclosed
EP-0772594-A1 IMINOXYCARBOXYLATES AND DERIVATIVES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS Abbott Laboratories (US) 1997-05-14 EP disclosed
US-5512581-A ANTIINFLAMMATORY AGENT ABBOTT LABORATORIES (US) 1996-04-30 US disclosed
WO-1996002507-A1 IMINOXYCARBOXYLATES AND DERIVATIVES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS ABBOTT LABORATORIES (US) 1996-02-01 WO disclosed
EP-0666849-A4 ARYL AND HETEROARYLMETHOXYPHENYL INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS. ABBOTT LAB (US) 1995-12-13 EP disclosed
EP-0666849-A1 ARYL AND HETEROARYLMETHOXYPHENYL INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS ABBOTT LABORATORIES (US) 1995-08-16 EP disclosed
US-5358955-A Antiinflammatory agents ABBOTT LABORATORIES (US) 1994-10-25 US disclosed
WO-1994010148-A1 ARYL AND HETEROARYLMETHOXYPHENYL INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS ABBOTT LABORATORIES (US) 1994-05-11 WO disclosed
EP-0344519-B1 SUBSTITUTED 4-(QUINOLIN-2-YL-METHOXY)PHENYL-ACETIC-ACID DERIVATIVES BAYER AG (DE) 1993-04-14 EP disclosed
US-4970215-A Substituted 4-(quinolin-2-yl-methoxy)phenyl-acetic acid derivatives and anti-allergic use thereof BAYER AKTIENGESELLSCHAFT (DE) 1990-11-13 US disclosed