SCHEMBL7752908

SCHEMBL7752908

O=C(c1ccccc1)c1ccc(F)c(Br)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.58
CYP1A2 P05177 1/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C19 P33261 1/20 0.58
ATM Q13315 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
ALDH1A1 P00352 2/20 0.52
SRD5A2 P31213 2/20 0.50
IDO1 P14902 1/20 0.50
TDO2 P48775 1/20 0.50
RAB9A P51151 4/20 0.47
NPC1 O15118 3/20 0.47
HSD17B14 Q9BPX1 1/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
PBRM1 Q86U86 1/20 0.47
ALOX15 P16050 2/20 0.47
TP53 P04637 1/20 0.47
TSHR P16473 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30817696 0.90 ALDH1A1 (0.52) HPGDCYP1A2CYP2D6CYP2C19ATM
SCHEMBL4784600 0.85 IDO1 (0.57) HPGDCYP1A2CYP2D6CYP2C19IDO1
SCHEMBL1129171 0.85 ATM (0.55) HPGDCYP1A2CYP2D6CYP2C19ATM
SCHEMBL27563858 0.82 HPGD (0.64) HPGDCYP1A2CYP2D6CYP2C19ATM
SCHEMBL332679 0.82 ATM (0.61) HPGDATMTDP1L3MBTL1ALDH1A1
SCHEMBL30391232 0.82 HPGD (0.64) HPGDCYP1A2CYP2D6CYP2C19ATM
SCHEMBL383767 0.81 MEN1 (0.57) HPGDCYP1A2CYP2D6CYP2C19TDP1
SCHEMBL104151 0.80 TTR (0.50) L3MBTL1SRD5A2IDO1TDO2RAB9A
SCHEMBL31302316 0.80 TTR (0.50) L3MBTL1SRD5A2IDO1TDO2RAB9A
SCHEMBL28635108 0.79 CYP1A2 (0.60) HPGDCYP1A2CYP2D6CYP2C19ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000031163-A2 POLY(ARYLENE ETHER) HOMOPOLYMER COMPOSITIONS AND METHODS OF MANUFACTURE THEREOF ALLIEDSIGNAL INC. (US) 2000-06-02 WO claimed
CN-116425782-A Preparation method of 5-acetyl-2-fluorobenzeneboronic acid pinacol ester 烟台盛凯伦化学科技有限公司 2023-07-14 CN disclosed
WO-2020253711-A1 PYRROLOPYRIDONE COMPOUND, PREPARATION METHOD THEREFOR, AND COMPOSITION AND USE THEREOF 中国科学院上海药物研究所 2020-12-24 WO disclosed
EP-1068255-A2 POLY(ARYLENE ETHER) COMPOSITIONS AND METHODS OF MANUFACTURE THEREOF AlliedSignal Inc. (US) 2001-01-17 EP disclosed
WO-2000031163-A2 POLY(ARYLENE ETHER) HOMOPOLYMER COMPOSITIONS AND METHODS OF MANUFACTURE THEREOF ALLIEDSIGNAL INC. (US) 2000-06-02 WO disclosed
WO-1999029761-A2 POLY(ARYLENE ETHER) COMPOSITIONS AND METHODS OF MANUFACTURE THEREOF ALLIEDSIGNAL INC. (US) 1999-06-17 WO disclosed