SCHEMBL7754941

SCHEMBL7754941

COc1cccc(S(=O)(=O)NCCC(=O)NC(Cc2cncn2C)c2ccc(C#N)c(F)c2)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 3/20 0.39
KDM4E B2RXH2 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
MEP1B Q16820 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.36
ATM Q13315 1/20 0.36
FNTA P49354 6/20 0.35
FNTB P49356 6/20 0.35
AKR1C3 P42330 1/20 0.34
S1PR3 Q99500 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PGGT1B P53609 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7754126 0.85 PTPRB (0.38) KDM4EFNTAFNTBS1PR3ALDH1A1
SCHEMBL7754946 0.84 L3MBTL1 (0.40) TRPV4MEP1BL3MBTL1ATMFNTA
Hydrochloric Acid SCHEMBL7757576 0.81 FNTA (0.39) FNTAFNTBS1PR3
SCHEMBL7220418 0.79 ALDH1A1 (0.40) TRPV4MEP1BL3MBTL1ATMFNTA
SCHEMBL7755612 0.77 FNTA (0.39) FNTAFNTBPGGT1B
SCHEMBL7220168 0.74 FNTA (0.37) TRPV4MEP1BL3MBTL1ATMFNTA
SCHEMBL8194917 0.72 FNTA (0.42) FNTAFNTB
SCHEMBL7755338 0.72 PTPRB (0.41) KDM4EFNTAFNTBALDH1A1PGGT1B
SCHEMBL7754130 0.69 FNTA (0.41) FNTAFNTBPGGT1B
SCHEMBL7681015 0.69 L3MBTL1 (0.39) TRPV4CYP2D6CYP2C19MEP1BL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001051126-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-07-19 WO disclosed