Acridan

Acridan

SCHEMBL7755741

CN1c2ccccc2C(C(=O)Oc2ccccc2)c2ccccc21.c1ccc2c(c1)Cc1ccccc1N2

nearest known ligand 0.42

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
EGFR P00533 2/20 0.37
SRC P12931 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
BRD4 O60885 1/20 0.36
CREBBP Q92793 1/20 0.36
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
SLC6A2 P23975 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
SLC6A4 P31645 1/20 0.35
ADRA1A P35348 1/20 0.35
HRH1 P35367 1/20 0.35
HTR2B P41595 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30132855 0.85 HDAC4 (0.55) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL2218308 0.85 HDAC4 (0.55) HDAC4HDAC7HDAC5EGFRSRC
Acridan SCHEMBL6342017 0.83 HDAC4 (0.38) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL13005780 0.81 HDAC4 (0.57) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL28319597 0.78 HDAC4 (0.48) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL7793810 0.77 HDAC4 (0.50) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL27487537 0.77 CYP1A2 (0.46) EGFRCYP1A2CYP2C9CYP2C19L3MBTL1
SCHEMBL2985418 0.76 HDAC4 (0.51) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL7796545 0.76 HDAC4 (0.51) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL3769074 0.76 HDAC4 (0.44) HDAC4HDAC7HDAC5EGFRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0755457-B1 Novel Aryl-N-Alkylacridanthiocarboxylate derivatives useful for chemiluminescent detection LUMIGEN INC (US) 2001-02-21 EP disclosed
EP-0755457-A4 NOVEL ARYL-N-ALKYLACRIDANTHIOCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN INC (US) 1997-07-16 EP disclosed
EP-0755457-A1 NOVEL ARYL-N-ALKYLACRIDANTHIOCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN, INC. (US) 1997-01-29 EP disclosed
US-5523212-A OXIDATION WITH PEROXIDE AND PEROXIDASE TO EXCITED ACRIDONE DERIVATIVE; DETECTING PROTEINS, HAPTENS, ANTIBODIES, ENZYMES LUMIGEN, INC. (US) 1996-06-04 US disclosed
WO-1995028495-A1 NOVEL ARYL-N-ALKYLACRIDANTHIOCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN, INC. (US) 1995-10-26 WO disclosed