SCHEMBL7756019

SCHEMBL7756019

CC(=O)C(=Cc1ccc(Cl)c(Cl)c1)C(C)=O

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
KDM4E B2RXH2 3/20 0.55
TDP1 Q9NUW8 2/20 0.54
GAA P10253 1/20 0.54
GLA P06280 1/20 0.52
POLB P06746 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
MAPT P10636 2/20 0.51
GLO1 Q04760 1/20 0.46
PYGL P06737 7/20 0.44
PTGS2 P35354 1/20 0.42
GUSB P08236 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28449048 0.87 GAA (0.50) ALDH1A1KDM4ETDP1GAAMAPT
SCHEMBL6137229 0.83 GLO1 (0.56) ALDH1A1KDM4ETDP1GAAPOLB
SCHEMBL6137225 0.83 GLO1 (0.56) ALDH1A1KDM4ETDP1GAAPOLB
SCHEMBL13792808 0.83 TDP1 (0.43) ALDH1A1KDM4ETDP1GAAGLA
SCHEMBL8038631 0.81 ALDH1A1 (0.47) ALDH1A1PYGLPTGS2
SCHEMBL7016901 0.80 TDP1 (0.46) ALDH1A1KDM4ETDP1GAAGLA
SCHEMBL7014950 0.80 TDP1 (0.46) ALDH1A1KDM4ETDP1GAAGLA
SCHEMBL14198040 0.79 ALDH1A1 (0.52) ALDH1A1PYGLPTGS2
SCHEMBL7615822 0.79 AKR1C3 (0.55) ALDH1A1PYGLPTGS2
SCHEMBL2008473 0.79 AKR1C3 (0.55) ALDH1A1PYGLPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001049660-A1 A PROCESS FOR PREPARING 3-{[3-CHLORO-4-(METHYLSULFONYL)-PHENYL]METHYLENE}-2,4-PENTANEDIONE ORION CORPORATION (FI) 2001-07-12 WO disclosed
EP-0440324-B1 Substituted beta-diketones and their use in the treatment of inflammatory bowel disease ORION YHTYMAE OY (FI) 2000-04-12 EP disclosed
US-5292771-A Treating inflammatory bowel disease ORION-YHTYMA OY (FI) 1994-03-08 US disclosed
US-5185370-A Substituted β-diketones and their use ORION-YHTYMA OY (FI) 1993-02-09 US disclosed
EP-0440324-A2 Substituted beta-diketones and their use ORION-YHTYMÀ„ OY (FI) 1991-08-07 EP disclosed