SCHEMBL7757057

SCHEMBL7757057

O=C(/C=C/c1ccc(O)cc1)c1c(O)c2ccccc2oc1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 7/20 1.00
MAPT P10636 4/20 0.76
KMT2A Q03164 4/20 0.76
KDM4E B2RXH2 3/20 0.76
RAB9A P51151 2/20 0.76
MEN1 O00255 2/20 0.76
RECQL P46063 1/20 0.76
GPR55 Q9Y2T6 1/20 0.76
CYP1A2 P05177 1/20 0.71
CYP2C9 P11712 1/20 0.71
CYP2C19 P33261 1/20 0.71
CA12 O43570 1/20 0.56
CA9 Q16790 1/20 0.56
LMNA P02545 2/20 0.50
HPGD P15428 1/20 0.50
ALDH1A1 P00352 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CYP3A4 P08684 2/20 0.49
HSPD1 P10809 1/20 0.49
PKM P14618 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7757059 1.00 NQO1 (1.00) NQO1MAPTKMT2AKDM4ERAB9A
SCHEMBL10362375 0.92 NQO1 (0.85) NQO1MAPTKMT2AKDM4ERAB9A
SCHEMBL10362376 0.92 NQO1 (0.85) NQO1MAPTKMT2AKDM4ERAB9A
SCHEMBL31419764 0.92 NQO1 (0.85) NQO1MAPTKMT2AKDM4ERAB9A
SCHEMBL13100090 0.90 NQO1 (0.81) NQO1MAPTKMT2AKDM4ERAB9A
SCHEMBL30214941 0.84 NQO1 (0.72) NQO1MAPTKMT2AKDM4ERAB9A
SCHEMBL30214865 0.82 NQO1 (0.69) NQO1MAPTKMT2AKDM4ERAB9A
SCHEMBL30933367 0.81 NQO1 (0.67) NQO1MAPTKMT2AKDM4ERAB9A
SCHEMBL27349811 0.81 NQO1 (0.67) NQO1MAPTKMT2AKDM4ERAB9A
SCHEMBL13403222 0.77 NQO1 (0.63) NQO1MAPTKMT2AKDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015183931-A1 STABILIZED CHEMILUMINESCENT SYSTEM LI-COR, INC. (US) 2015-12-03 WO claimed
US-20150346202-A1 STABILIZED CHEMILUMINESCENT SYSTEM Ll-COR, INC. (US) 2015-12-03 US claimed
US-10036708-B2 Solution phase homogeneous assays BECKMAN COULTER, INC. (US) 2018-07-31 US disclosed
US-10036708-B2 Solution phase homogeneous assays BECKMAN COULTER, INC. (US) 2018-07-31 US disclosed
EP-2401392-B1 SOLUTION PHASE HOMOGENEOUS ASSAYS BECKMAN COULTER INC (US) 2017-01-25 EP disclosed
WO-2015183931-A1 STABILIZED CHEMILUMINESCENT SYSTEM LI-COR, INC. (US) 2015-12-03 WO disclosed
US-20150346202-A1 STABILIZED CHEMILUMINESCENT SYSTEM Ll-COR, INC. (US) 2015-12-03 US disclosed
US-20150212005-A1 SOLUTION PHASE HOMOGENEOUS ASSAYS BECKMAN COULTER, INC. 2015-07-30 US disclosed
US-20150212005-A1 SOLUTION PHASE HOMOGENEOUS ASSAYS BECKMAN COULTER, INC. 2015-07-30 US disclosed
US-9029092-B2 Solution phase homogeneous assays BECKMAN COULTER, INC. (US) 2015-05-12 US disclosed
US-9029092-B2 Solution phase homogeneous assays BECKMAN COULTER, INC. (US) 2015-05-12 US disclosed
US-20100267071-A1 SOLUTION PHASE HOMOGENEOUS ASSAYS BECKMAN COULTER, INC. (US) 2010-10-21 US disclosed
US-20100267071-A1 SOLUTION PHASE HOMOGENEOUS ASSAYS BECKMAN COULTER, INC. (US) 2010-10-21 US disclosed
WO-2010099479-A1 NON SEPARATION ASSAYS WITH SELECTIVE SIGNAL INHIBITORS BECKMAN COULTER, INC. (US) 2010-09-02 WO disclosed
WO-2010099486-A1 SOLUTION PHASE HOMOGENEOUS ASSAYS BECKMAN COULTER, INC. (US) 2010-09-02 WO disclosed
EP-0755457-B1 Novel Aryl-N-Alkylacridanthiocarboxylate derivatives useful for chemiluminescent detection LUMIGEN INC (US) 2001-02-21 EP disclosed
WO-1999001768-A1 PEROXIDASE-CATALYSED FLUORESCENCE NYCOMED AMERSHAM PLC (GB) 1999-01-14 WO disclosed
US-5523212-A OXIDATION WITH PEROXIDE AND PEROXIDASE TO EXCITED ACRIDONE DERIVATIVE; DETECTING PROTEINS, HAPTENS, ANTIBODIES, ENZYMES LUMIGEN, INC. (US) 1996-06-04 US disclosed
WO-1995023971-A1 NOVEL ARYL N-ALKYLACRIDANCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN, INC. (US) 1995-09-08 WO disclosed