SCHEMBL7757934

SCHEMBL7757934

COc1ccc(CN2CCN(C(C)C)CC2)c(OC(=O)c2ccccc2)c1OC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
HTT P42858 2/20 0.56
CYP2C19 P33261 1/20 0.54
MEN1 O00255 5/20 0.52
KMT2A Q03164 5/20 0.52
KDM4E B2RXH2 4/20 0.50
CHRM2 P08172 2/20 0.49
OPRK1 P41145 2/20 0.49
LMNA P02545 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
CHRM1 P11229 1/20 0.49
DRD2 P14416 1/20 0.49
ADRA2B P18089 1/20 0.49
ADRA2C P18825 1/20 0.49
CNR1 P21554 1/20 0.49
SLC6A2 P23975 1/20 0.49
HTR2A P28223 1/20 0.49
HTR2C P28335 1/20 0.49
ADRA1A P35348 1/20 0.49
HRH1 P35367 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8640153 0.99 ALDH1A1 (0.55) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL7757458 0.90 HTT (0.61) ALDH1A1HTTCYP2C19MEN1KMT2A
Hydrochloric Acid SCHEMBL8637261 0.89 HTT (0.60) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL7758476 0.88 ALDH1A1 (0.59) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL7758568 0.88 MEN1 (0.64) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL7756417 0.88 ALDH1A1 (0.59) ALDH1A1HTTCYP2C19MEN1KMT2A
Hydrochloric Acid SCHEMBL8635524 0.87 ALDH1A1 (0.58) ALDH1A1HTTCYP2C19MEN1KMT2A
Hydrochloric Acid SCHEMBL8642718 0.87 ALDH1A1 (0.58) ALDH1A1HTTCYP2C19MEN1KMT2A
Hydrochloric Acid SCHEMBL8639585 0.87 MEN1 (0.62) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL7753771 0.86 ALDH1A1 (0.57) ALDH1A1HTTCYP2C19MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0847999-B1 N-benzylpiperazine derivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-03-21 EP disclosed
EP-0847999-A1 N-benzylpiperazine derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1998-06-17 EP disclosed