SCHEMBL7761646

SCHEMBL7761646

Oc1c(-c2ccccc2)c(C(F)(F)F)nc2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ENPP1 P22413 4/20 0.51
ESR1 P03372 5/20 0.43
DHODH Q02127 2/20 0.41
PDE10A Q9Y233 1/20 0.41
LMNA P02545 1/20 0.41
ESR2 Q92731 3/20 0.40
KDM4E B2RXH2 2/20 0.40
MAPT P10636 1/20 0.40
GYS1 P13807 1/20 0.40
POLB P06746 2/20 0.40
DCTPP1 Q9H773 1/20 0.39
BACE1 P56817 1/20 0.39
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15647912 0.82 RXFP1 (0.47) ENPP1KDM4EMAPTPOLBALDH1A1
SCHEMBL15648268 0.82 ENPP1 (0.42) ENPP1ESR1DHODHLMNAESR2
SCHEMBL16632042 0.80 ENPP1 (0.67) ENPP1ESR1ESR2KDM4EMAPT
SCHEMBL2788828 0.79 KDM4E (0.42) LMNAKDM4EMAPTPOLBDCTPP1
SCHEMBL625364 0.77 LMNA (0.46) ESR1DHODHPDE10ALMNAESR2
SCHEMBL28027243 0.77 ENPP1 (0.48) ENPP1ESR1ESR2KDM4EMAPT
SCHEMBL394890 0.75 DHODH (0.50) DHODHPDE10ALMNAKDM4EPOLB
SCHEMBL624087 0.75 LMNA (0.45) ESR1DHODHPDE10ALMNAESR2
SCHEMBL12693813 0.74 ERN1 (0.53) LMNAKDM4EMAPTPOLBDCTPP1
SCHEMBL11375363 0.74 GAA (0.46) DHODHPDE10ALMNAKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105829295-A Phenyl Linked Quinolinyl Modulators Of Ror-Gamma-T 詹森药业有限公司 2016-08-03 CN disclosed
CN-105073729-A Phenyl-linked quinolinyl modulators of ROR γ t JANSSEN PHARMACEUTICA NV 2015-11-18 CN disclosed
EP-1087790-A2 USE OF A COMPOUND HAVING AFFINITY FOR THE BENZODIAZEPINE MITOCHONDRIAL RECEPTOR IN CANCER THERAPY CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2001-04-04 EP disclosed
WO-1999066958-A2 USE OF A COMPOUND HAVING AFFINITY FOR THE BENZODIAZEPINE MITOCHONDRIAL RECEPTOR IN CANCER THERAPY CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 1999-12-29 WO disclosed