SCHEMBL7763004

SCHEMBL7763004

Oc1ccc2ncnc(Nc3ccc(F)c(F)c3)c2c1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 2/20 0.60
EGFR P00533 9/20 0.57
RAF1 P04049 5/20 0.57
BRAF P15056 5/20 0.57
ERBB2 P04626 1/20 0.56
DYRK1A Q13627 1/20 0.55
RIPK2 O43353 1/20 0.54
RET P07949 1/20 0.54
KIF5B P33176 1/20 0.54
KDR P35968 1/20 0.54
NOD1 Q9Y239 1/20 0.54
ABCG2 Q9UNQ0 1/20 0.54
GLA P06280 1/20 0.53
HTT P42858 1/20 0.53
GAA P10253 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL641359 0.88 EGFR (0.75) EGFRRAF1BRAFERBB2KDR
Hydrochloric Acid SCHEMBL7760887 0.83 EGFR (0.76) EGFRERBB2DYRK1A
SCHEMBL13599953 0.80 RAF1 (0.79) ALKEGFRRAF1BRAFERBB2
SCHEMBL4738585 0.80 EGFR (0.80) EGFRRAF1BRAFERBB2GLA
SCHEMBL8104967 0.78 EGFR (0.57) EGFRERBB2DYRK1A
SCHEMBL7766632 0.78 EGFR (0.57) EGFRRAF1BRAFERBB2RIPK2
Hydrochloric Acid SCHEMBL7763512 0.77 ALK (0.69) ALKEGFRNOD1ABCG2HTT
SCHEMBL9478 0.77 EGFR (0.77) ALKEGFRRAF1BRAFERBB2
Hydrochloric Acid SCHEMBL8104687 0.77 EGFR (0.70) EGFRERBB2
SCHEMBL3664557 0.77 EGFR (0.81) ALKEGFRRAF1BRAFERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0824525-B1 QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2001-06-13 EP disclosed
US-5932574-A ANTICANCER AGENT ZENECA LIMITED (GB) 1999-08-03 US disclosed
EP-0824525-A1 QUINAZOLINE DERIVATIVES ZENECA LIMITED (GB) 1998-02-25 EP disclosed
WO-1996033977-A1 QUINAZOLINE DERIVATIVES ZENECA LIMITED (GB) 1996-10-31 WO disclosed