SCHEMBL7764986

SCHEMBL7764986

C/C(=C\c1ccccc1-c1ccccc1/C=C(\C)C(=O)O)C(=O)O

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.61
APEX1 P27695 8/20 0.54
HTT P42858 1/20 0.42
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
NR4A2 P43354 1/20 0.41
RXRG P48443 1/20 0.41
KDM4E B2RXH2 1/20 0.41
LTB4R Q15722 1/20 0.40
LTB4R2 Q9NPC1 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7764991 1.00 AKR1C3 (0.61) AKR1C3APEX1HTTRXRARXRB
SCHEMBL22042820 0.91 AKR1C3 (0.52) AKR1C3APEX1RXRARXRBNR4A2
SCHEMBL240897 0.90 AKR1C3 (0.55) AKR1C3APEX1RXRARXRBNR4A2
SCHEMBL5852799 0.90 AKR1C3 (0.55) AKR1C3APEX1RXRARXRBNR4A2
SCHEMBL3893886 0.89 AKR1C3 (0.68) AKR1C3APEX1HTTRXRARXRB
SCHEMBL8746671 0.89 AKR1C3 (0.68) AKR1C3APEX1HTTRXRARXRB
SCHEMBL31666241 0.89 AKR1C3 (0.68) AKR1C3APEX1HTTRXRARXRB
SCHEMBL22042826 0.84 APEX1 (0.49) AKR1C3APEX1RXRARXRBNR4A2
SCHEMBL208434 0.82 AKR1C3 (0.59) AKR1C3APEX1
SCHEMBL11783107 0.82 AKR1C3 (0.59) AKR1C3APEX1HTTRXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001087829-A1 BISACYLGUANIDINE MERCK PATENT GMBH (DE) 2001-11-22 WO disclosed