SCHEMBL7765015

SCHEMBL7765015

C/C(=C\c1ccccc1C(=O)c1ccccc1/C=C(\C)C(=O)O)C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.57
APEX1 P27695 8/20 0.44
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
NR4A2 P43354 1/20 0.40
RXRG P48443 1/20 0.40
KDM4E B2RXH2 1/20 0.40
HTT P42858 1/20 0.40
ALDH1A1 P00352 2/20 0.38
TP53 P04637 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
TSHR P16473 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
DHODH Q02127 1/20 0.38
TRPM8 Q7Z2W7 1/20 0.38
ALOX15 P16050 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7765021 1.00 AKR1C3 (0.57) AKR1C3APEX1RXRARXRBNR4A2
SCHEMBL474960 0.91 AKR1C3 (0.52) AKR1C3APEX1ALDH1A1GAAMAPT
SCHEMBL31666241 0.86 AKR1C3 (0.68) AKR1C3APEX1RXRARXRBNR4A2
SCHEMBL8746671 0.86 AKR1C3 (0.68) AKR1C3APEX1RXRARXRBNR4A2
SCHEMBL3893886 0.86 AKR1C3 (0.68) AKR1C3APEX1RXRARXRBNR4A2
SCHEMBL7764223 0.85 AKR1C3 (0.59) AKR1C3APEX1HTTALDH1A1GAA
SCHEMBL7764230 0.85 AKR1C3 (0.59) AKR1C3APEX1HTTALDH1A1GAA
SCHEMBL2954153 0.82 AKR1C3 (0.50) AKR1C3APEX1CYP2C9
SCHEMBL7764991 0.80 AKR1C3 (0.61) AKR1C3APEX1RXRARXRBNR4A2
SCHEMBL7764986 0.80 AKR1C3 (0.61) AKR1C3APEX1RXRARXRBNR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001087829-A1 BISACYLGUANIDINE MERCK PATENT GMBH (DE) 2001-11-22 WO disclosed