SCHEMBL7765079

SCHEMBL7765079

CCOC(=O)c1ccc(OCC)cc1C(=O)OCC

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.58
KDM4E B2RXH2 6/20 0.54
CA12 O43570 2/20 0.53
CA1 P00915 2/20 0.53
CA2 P00918 2/20 0.53
CA7 P43166 2/20 0.53
CA9 Q16790 2/20 0.53
CA14 Q9ULX7 2/20 0.53
ALDH1A1 P00352 8/20 0.52
PKM P14618 1/20 0.52
MAPT P10636 4/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
NPSR1 Q6W5P4 1/20 0.49
LMNA P02545 3/20 0.48
NPC1 O15118 2/20 0.48
TDP1 Q9NUW8 2/20 0.48
GAA P10253 2/20 0.48
HTT P42858 1/20 0.48
HPGD P15428 4/20 0.47
HSD17B10 Q99714 4/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8142570 0.88 TSHR (0.53) TSHRKDM4ECA12CA1CA2
SCHEMBL9541238 0.88 KDM4E (0.53) TSHRKDM4ECA12CA1CA2
SCHEMBL9952719 0.86 CA12 (0.73) TSHRKDM4ECA12CA1CA2
SCHEMBL10469566 0.86 CA12 (0.68) TSHRKDM4ECA12CA1CA2
SCHEMBL3999898 0.86 KDM4E (0.55) TSHRKDM4ECA12CA1CA2
SCHEMBL21543853 0.86 TDP1 (0.55) KDM4ECA12CA1CA2CA7
SCHEMBL28275232 0.86 HPGD (0.60) TSHRKDM4ECA12CA1CA2
SCHEMBL13366219 0.85 KDM4E (0.50) TSHRKDM4ECA12CA1CA2
SCHEMBL22749335 0.85 ALDH1A1 (0.58) TSHRKDM4ECA12CA1CA2
SCHEMBL31225318 0.85 KDM4E (0.50) TSHRKDM4ECA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825178-B1 Phenyl-substituted alkenoylguanidides, process for their preparation, their use as drugs or in diagnostic agents and drugs containing them HOECHST AG (DE) 2001-06-20 EP disclosed
US-6005010-A CARDIOVASCULAR DISORDERS, ANTIARRHYTHMIA AGENTS AND ANTIISCHEMIC AGENTS HOECHST AKTIENGESELLSCHAFT (DE) 1999-12-21 US disclosed
EP-0825178-A1 Phenyl-substituted alkenoylguanidides, process for their preparation, their use as drugs or in diagnostic agents and drugs containing them HOECHST AKTIENGESELLSCHAFT (DE) 1998-02-25 EP disclosed