SCHEMBL7765338

SCHEMBL7765338

O=c1[nH]c(N(I)Cc2ccccc2)nc2nc[nH]c12

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PNP P00491 2/20 0.46
PDE5A O76074 1/20 0.43
GRIA1 P42261 1/20 0.43
GRIA2 P42262 1/20 0.43
GRIA3 P42263 1/20 0.43
GRIA4 P48058 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3433603 0.88 TSHR (0.52) PNPPDE5AGRIA1GRIA2GRIA3
SCHEMBL3425179 0.86 PNP (0.48) PNPPDE5AGRIA1GRIA2GRIA3
SCHEMBL1533594 0.86 PNP (0.44) PNPPDE5AGRIA1GRIA2GRIA3
SCHEMBL5798037 0.86 GRIA1 (0.45) PNPPDE5AGRIA1GRIA2GRIA3
SCHEMBL2776930 0.84 PNP (0.46) PNPPDE5AGRIA1GRIA2GRIA3
SCHEMBL30080348 0.84 PDE5A (0.43) PNPPDE5AGRIA1GRIA2GRIA3
SCHEMBL30248422 0.82 CYP1A2 (0.47) PNPPDE5AGRIA1GRIA2GRIA3
SCHEMBL1286929 0.78 PNP (0.50) PNPPDE5AGRIA1GRIA2GRIA3
SCHEMBL29131184 0.77 PNP (0.43) PNPPDE5AGRIA1GRIA2GRIA3
SCHEMBL5084818 0.75 PNP (0.58) PNPPDE5AGRIA1GRIA2GRIA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001085221-A2 ASSESSING LEVELS OF O6-ALKYLGUANINE-DNA ALKYLTRANSFERASE IN VIVO DUKE UNIVERSITY (US) 2001-11-15 WO disclosed