SCHEMBL7765693

SCHEMBL7765693

OCc1c(Cl)cccc1Oc1ccccc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.69
LMNA P02545 2/20 0.57
MAPT P10636 2/20 0.54
POLB P06746 1/20 0.54
FABP3 P05413 1/20 0.51
FABP4 P15090 1/20 0.51
L3MBTL1 Q9Y468 2/20 0.49
GAA P10253 1/20 0.49
SMOX Q9NWM0 2/20 0.48
KDM1A O60341 1/20 0.48
RCOR1 Q9UKL0 1/20 0.48
ALDH1A1 P00352 3/20 0.48
NPSR1 Q6W5P4 1/20 0.48
TTR P02766 1/20 0.46
MAPK8 P45983 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
LTA4H P09960 1/20 0.46
KMT2A Q03164 1/20 0.45
RHEB Q15382 2/20 0.43
AKR1B1 P15121 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14382784 0.81 DPP4 (0.69) DPP4LMNAMAPTPOLBFABP3
SCHEMBL1191734 0.81 DPP4 (0.69) DPP4LMNAMAPTPOLBFABP3
SCHEMBL112755 0.81 DPP4 (1.00) DPP4LMNAMAPTPOLBFABP3
SCHEMBL25942519 0.80 EPAS1 (0.46) DPP4LMNAMAPTPOLBL3MBTL1
SCHEMBL14097997 0.80 LMNA (0.46) DPP4LMNAMAPTPOLBL3MBTL1
SCHEMBL16245360 0.79 HRH1 (0.50) DPP4LMNAL3MBTL1GAAALDH1A1
SCHEMBL3790160 0.78 DPP4 (0.62) DPP4LMNAMAPTPOLBL3MBTL1
SCHEMBL14452021 0.77 DPP4 (0.63) DPP4LMNAMAPTPOLBFABP3
SCHEMBL7769554 0.77 DPP4 (0.63) DPP4LMNAMAPTPOLBFABP3
SCHEMBL11500020 0.77 DPP4 (0.63) DPP4LMNAMAPTPOLBFABP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1216052-C Anti-neurodegeneratively active 10-aminoaliphatyl-dibenz (b,f) oxepines NAVARTIS AG (CH) 2005-08-24 CN disclosed
EP-0726265-B1 10-Aminoaliphatyl-dibenz(b,f)oxepins with antineurodegenarative activity NOVARTIS AG (CH) 2001-07-25 EP disclosed
US-5780501-A ADMINISTERING TO A MAMMAL NOVARTIS CORPORATION (US) 1998-07-14 US disclosed
US-5780500-A Anti-neurodegeneratively active 10-aminoaliphatyl-dibenzi b,f! oxepines NOVARTIS CORPORATION (US) 1998-07-14 US disclosed
CN-1137039-A Anti-neurodegeneratively active 10-aminoaliphatyl-dibenz (b,f) oxepines CIBA GEIGY AG (CH) 1996-12-04 CN disclosed
EP-0726265-A1 10-Aminoaliphatyl-dibenz(b,f)oxepins with antineurodegenarative activity CIBA-GEIGY AG (CH) 1996-08-14 EP disclosed