SCHEMBL7767206

SCHEMBL7767206

CCO/C(=C(\C#N)c1cccc(Cl)c1Cl)C(OCC)OCC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
TAS1R2 Q8TE23 1/20 0.38
TSHR P16473 3/20 0.34
ALDH1A1 P00352 3/20 0.34
LMNA P02545 3/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HTT P42858 1/20 0.33
CASP1 P29466 1/20 0.33
MAPT P10636 2/20 0.33
METTL3 Q86U44 1/20 0.33
SLC6A3 Q01959 3/20 0.32
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
KCNH2 Q12809 1/20 0.32
ERCC5 P28715 1/20 0.32
FEN1 P39748 1/20 0.32
CYP2C9 P11712 3/20 0.32
KDM4E B2RXH2 2/20 0.32
MEN1 O00255 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7767210 1.00 TAS1R3 (0.38) TAS1R3TAS1R1TAS1R2TSHRALDH1A1
SCHEMBL310647 0.78 TAS1R3 (0.37) TAS1R3TAS1R1TAS1R2TSHRALDH1A1
SCHEMBL310648 0.78 TAS1R3 (0.37) TAS1R3TAS1R1TAS1R2TSHRALDH1A1
SCHEMBL5070752 0.69 TAS1R3 (0.38) TAS1R3TAS1R1TAS1R2TSHRALDH1A1
SCHEMBL5070753 0.69 TAS1R3 (0.38) TAS1R3TAS1R1TAS1R2TSHRALDH1A1
SCHEMBL1554603 0.68 GPR35 (0.42) TAS1R3TAS1R1TAS1R2TSHRALDH1A1
SCHEMBL1554601 0.68 GPR35 (0.42) TAS1R3TAS1R1TAS1R2TSHRALDH1A1
SCHEMBL10665640 0.67 TSHR (0.44) TAS1R3TAS1R1TAS1R2TSHRALDH1A1
SCHEMBL11418791 0.67 TSHR (0.63) TAS1R3TAS1R1TAS1R2TSHRALDH1A1
SCHEMBL7772728 0.67 TSHR (0.44) TAS1R3TAS1R1TAS1R2TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0879230-B1 OPTICALLY ACTIVE PHENYL PYRIMIDINE DERIVATIVE AS ANALGESIC AGENT GLAXO GROUP LTD (GB) 2001-07-25 EP disclosed
US-6124308-A ANALGESICS, ANTICONVULSANTS, TREATING IRRITABLE BOWEL SYNDROME OR BIPOLAR DISORDER GLAXO WELLCOME INC. (US) 2000-09-26 US disclosed