SCHEMBL7767398

SCHEMBL7767398

O=c1[nH]c2ccc(CCl)cc2s1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.50
PDE3A Q14432 2/20 0.50
PGR P06401 2/20 0.49
CMA1 P23946 1/20 0.49
HTR1A P08908 7/20 0.47
HTR2C P28335 6/20 0.47
MAPT P10636 1/20 0.46
DRD2 P14416 1/20 0.40
HTR2A P28223 1/20 0.40
ALDH1A1 P00352 1/20 0.39
PKM P14618 1/20 0.39
KIF11 P52732 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17080919 0.86 HTR1A (0.51) PDE3BPDE3APGRCMA1HTR1A
SCHEMBL1325447 0.83 HTR1A (0.49) PDE3BPDE3APGRCMA1HTR1A
SCHEMBL9684052 0.82 HTR1A (0.48) PDE3BPDE3APGRCMA1HTR1A
SCHEMBL9204486 0.81 MAPT (0.59) PDE3BPDE3APGRCMA1HTR1A
SCHEMBL7765507 0.81 PDE3B (0.50) PDE3BPDE3APGRCMA1HTR1A
SCHEMBL9685648 0.80 CMA1 (0.56) PDE3BPDE3APGRCMA1HTR1A
SCHEMBL9992658 0.80 PDE3B (0.49) PDE3BPDE3APGRCMA1HTR1A
SCHEMBL4882695 0.79 HTR1A (0.51) PDE3BPDE3APGRCMA1HTR1A
SCHEMBL9684901 0.79 PDE3B (0.51) PDE3BPDE3APGRCMA1HTR1A
SCHEMBL7332557 0.79 HTR1A (0.51) PDE3BPDE3APGRCMA1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1072655-C New heterocyclic aminomethyl compounds, process for preparing them and pharmaceutical compositions containing them ADIR (FR) 2001-10-10 CN disclosed
EP-0841330-B1 Aminomethyl heterocyclic derivatives, process of their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-06-27 EP disclosed
US-5919784-A ANXIETY, DEPRESSION ADIR ET COMPAGNIE (FR) 1999-07-06 US disclosed
CN-1182083-A New heterocyclic aminomethyl compounds, process for preparing them and pharmaceutical compositions containing them ADIR (FR) 1998-05-20 CN disclosed
EP-0841330-A1 Aminomethyl heterocyclic derivatives, process of their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1998-05-13 EP disclosed