SCHEMBL7768166

SCHEMBL7768166

CNC(=O)c1cccc(OCCNCCCCC(=O)NCC(C)(C)C)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.47
KDM4E B2RXH2 2/20 0.43
HDAC3 O15379 1/20 0.43
KMT2A Q03164 3/20 0.43
HPGD P15428 2/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 2/20 0.43
GAA P10253 1/20 0.43
SMPD1 P17405 3/20 0.42
HTT P42858 1/20 0.41
SCN9A Q15858 1/20 0.41
DRD2 P14416 2/20 0.40
DRD4 P21917 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40
F10 P00742 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7768178 0.82 MAPT (0.57) MAOBKMT2AMEN1ALDH1A1
SCHEMBL7764594 0.81 MAPT (0.46) MAOBKDM4EKMT2AHPGDMEN1
SCHEMBL7772444 0.81 MAPT (0.46) MAOBKDM4EHDAC3KMT2AHPGD
SCHEMBL7768170 0.79 ALDH1A1 (0.47) KDM4EHDAC3KMT2AHPGDMEN1
SCHEMBL7769386 0.74 ALDH1A1 (0.53) KMT2AHPGDALDH1A1DRD2DRD4
SCHEMBL7565657 0.73 HTR1A (0.45) KDM4EHDAC3KMT2AHPGDMEN1
SCHEMBL25974208 0.72 HDAC8 (0.50) KMT2AHPGDALDH1A1SMPD1HTT
SCHEMBL24500604 0.72 SMPD1 (0.70) KMT2AMEN1ALDH1A1SMPD1MAPK1
SCHEMBL7567224 0.71 POLB (0.48) KDM4EHDAC3KMT2AMEN1ALDH1A1
SCHEMBL7768489 0.71 HDAC3 (0.43) KDM4EHDAC3KMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929515-B1 NOVEL PHENOXYETHYLAMINE DERIVATIVES, METHOD OF PREPARATION, APPLICATION AS MEDICINE AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME CONSEILS DE RECH S SOC D (FR) 2001-06-20 EP claimed
US-5998666-A ANTIULCER, ANTISECRETORY AGENTS; ANTIEMITIC SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (FR) 1999-12-07 US claimed
EP-0929515-A1 NOVEL PHENOXYETHYLAMINE DERIVATIVES, METHOD OF PREPARATION, APPLICATION AS MEDICINE AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 1999-07-21 EP claimed
WO-1998013337-A1 NOVEL PHENOXYETHYLAMINE DERIVATIVES, METHOD OF PREPARATION, APPLICATION AS MEDICINE AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 1998-04-02 WO claimed