SCHEMBL7768814

SCHEMBL7768814

COc1ccc(CC(SNC(=O)[C@@H](C)NC(=O)[C@@H]2CSCN2C(=O)C(C)(C)O)C2CCCCC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 1/20 0.39
ALDH1A1 P00352 3/20 0.35
PSMB8 P28062 5/20 0.35
PSMB5 P28074 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
BIRC2 Q13490 1/20 0.35
CHRM3 P20309 1/20 0.35
PSMB10 P40306 3/20 0.35
PSMB9 P28065 2/20 0.35
EPHX2 P34913 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ACACB O00763 1/20 0.35
PSMB2 P49721 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7110901 0.91 MEN1 (0.43) CACNA1BALDH1A1PSMB8PSMB5MEN1
SCHEMBL7105591 0.91 MEN1 (0.43) CACNA1BALDH1A1PSMB8PSMB5MEN1
SCHEMBL7110470 0.91 MEN1 (0.43) CACNA1BALDH1A1PSMB8PSMB5MEN1
SCHEMBL7772818 0.89 CACNA1B (0.39) CACNA1BALDH1A1PSMB8PSMB5BIRC2
SCHEMBL7768801 0.87 CACNA1B (0.39) CACNA1BALDH1A1PSMB8PSMB5BIRC2
SCHEMBL7774825 0.86 CACNA1B (0.44) CACNA1BALDH1A1PSMB8PSMB5BIRC2
SCHEMBL7105628 0.86 MEN1 (0.45) CACNA1BALDH1A1PSMB8PSMB5MEN1
SCHEMBL7110494 0.83 CACNA1B (0.50) CACNA1BMEN1KMT2ABIRC2
SCHEMBL7768808 0.82 CACNA1B (0.47) CACNA1BPSMB8PSMB5BIRC2PSMB9
SCHEMBL7111673 0.81 YAP1 (0.46) CACNA1BPSMB8PSMB5PSMB10PSMB9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1097929-A1 AMINO ACID DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2001-05-09 EP claimed
EP-1097929-A1 AMINO ACID DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2001-05-09 EP disclosed