SCHEMBL7770375

SCHEMBL7770375

CC(C)(C)[Si](C)(C)Cl.CC(C)(C)[Si](C)(C)O[C@H](CCc1cccnc1)COc1ccc(Br)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.36
TDP1 Q9NUW8 2/20 0.36
TP53 P04637 1/20 0.36
POLB P06746 1/20 0.36
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
PTAFR P25105 2/20 0.34
CHRNA7 P36544 2/20 0.34
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C9 P11712 2/20 0.33
MAPK1 P28482 2/20 0.33
LMNA P02545 1/20 0.33
KDM4E B2RXH2 2/20 0.32
GAA P10253 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
L3MBTL1 Q9Y468 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7773936 0.96 ALDH1A1 (0.36) ALDH1A1TDP1TP53POLBMEN1
SCHEMBL7774645 0.96 ALDH1A1 (0.36) ALDH1A1TDP1TP53POLBMEN1
SCHEMBL8551128 0.94 MEN1 (0.35) ALDH1A1TDP1TP53POLBMEN1
SCHEMBL7766506 0.85 ALDH1A1 (0.36) ALDH1A1TDP1TP53POLBMEN1
SCHEMBL7774215 0.84 GRM2 (0.34) ALDH1A1POLBMEN1KMT2ANPC1
SCHEMBL7766502 0.84 MEN1 (0.37) ALDH1A1TDP1TP53POLBMEN1
SCHEMBL7771572 0.84 MEN1 (0.37) ALDH1A1TDP1TP53POLBMEN1
SCHEMBL8117388 0.83 P2RX7 (0.36) ALDH1A1MEN1KMT2ACYP3A4LMNA
SCHEMBL7771575 0.82 MEN1 (0.39) ALDH1A1MEN1KMT2ACYP2D6MAPK1
SCHEMBL7766496 0.82 MEN1 (0.39) ALDH1A1MEN1KMT2ACYP2D6MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115706-A1 NOVEL COMPOUNDS AstraZeneca AB (SE) 2001-07-18 EP disclosed
EP-1115401-A1 NOVEL COMPOUNDS AstraZeneca AB (SE) 2001-07-18 EP disclosed
EP-1019375-A1 NOVEL PYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Astra Pharmaceuticals Limited (GB) 2000-07-19 EP disclosed
WO-2000018730-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2000-04-06 WO disclosed
WO-2000018731-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2000-04-06 WO disclosed
WO-1998042669-A1 NOVEL PYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ASTRA PHARMACEUTICALS LTD. (GB) 1998-10-01 WO disclosed