SCHEMBL7772092

SCHEMBL7772092

COc1cc(OCCN2CCCC2)cc(-c2ccc(OCCN3CCCC3)cc2)c1C(=O)c1csc2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 16/20 0.56
ESR2 Q92731 16/20 0.56
F2 P00734 1/20 0.48
KCNH2 Q12809 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
HSD17B10 Q99714 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7452470 0.89 ESR1 (0.49) ESR1ESR2F2KCNH2HRH3
SCHEMBL7414836 0.85 ESR1 (0.58) ESR1ESR2F2ALDH1A1CYP1A2
SCHEMBL7452427 0.85 ESR1 (0.51) ESR1ESR2F2ALDH1A1CYP1A2
SCHEMBL7445743 0.84 ESR1 (0.59) ESR1ESR2F2ALDH1A1CYP1A2
SCHEMBL8632802 0.84 MAPT (0.43) ESR1ESR2CYP1A2CYP2D6
SCHEMBL8635922 0.84 MAPT (0.43) ESR1ESR2CYP1A2CYP2D6
SCHEMBL7451880 0.82 HRH3 (0.51) ESR1ESR2F2KCNH2HRH3
SCHEMBL8634790 0.81 MAPT (0.48) ALDH1A1CYP1A2CYP2D6HSD17B10
SCHEMBL7445232 0.81 ESR1 (0.57) ESR1ESR2KCNH2ALDH1A1CYP1A2
SCHEMBL8642388 0.81 ESR1 (0.55) ESR1ESR2KCNH2ALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251921-B1 ADMINISTERING THROMBIN INHIBITING DIAMINE COMPOUND TO MAMMAL ELI LILLY AND COMPANY 2001-06-26 US disclosed