SCHEMBL7773194

SCHEMBL7773194

NC(CN1CCN(Cc2ccc(Cl)cc2)CC1)c1nc2ccc(F)cc2s1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.44
DRD2 P14416 3/20 0.44
CACNA1G O43497 1/20 0.43
MAPT P10636 1/20 0.43
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
LRRK2 Q5S007 1/20 0.39
ALDH1A1 P00352 1/20 0.39
AXL P30530 1/20 0.39
GFER P55789 1/20 0.39
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR1A P08908 1/20 0.38
HTR3A P46098 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
DRD4 P21917 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL7773390 0.99 KCNH2 (0.43) KCNH2DRD2CACNA1GMAPTNPC1
SCHEMBL27565702 0.95 DRD2 (0.49) KCNH2DRD2MAPTNPC1RAB9A
SCHEMBL7769219 0.90 NPC1 (0.45) KCNH2DRD2MAPTNPC1RAB9A
Fumaric Acid SCHEMBL7776854 0.83 ALDH1A1 (0.42) MAPTNPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL7775455 0.81 NPC1 (0.44) MAPTNPC1RAB9ASMN1; SMN2LRRK2
Bromide SCHEMBL7857770 0.81 NPC1 (0.44) MAPTNPC1RAB9ASMN1; SMN2LRRK2
SCHEMBL7773197 0.80 KCNH2 (0.43) KCNH2DRD2CACNA1GMAPTNPC1
SCHEMBL27565726 0.80 NPC1 (0.44) MAPTNPC1RAB9ASMN1; SMN2LRRK2
Bromide SCHEMBL7773393 0.79 KCNH2 (0.43) KCNH2DRD2CACNA1GMAPTNPC1
SCHEMBL7773430 0.79 CSNK1D (0.46) DRD2MAPTALDH1A1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1117663-A2 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 2001-07-25 EP disclosed
WO-2000018767-A9 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORP (US) 2001-04-19 WO disclosed
WO-2000018767-A2 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 2000-04-06 WO disclosed