SCHEMBL7773399

SCHEMBL7773399

NC(Cc1nc2ccccc2s1)N1CCN(c2ncc(F)cn2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.48
DRD3 P35462 8/20 0.48
DRD4 P21917 7/20 0.48
HTR7 P34969 6/20 0.48
HTR1A P08908 6/20 0.48
SIGMAR1 Q99720 3/20 0.48
ADRA2A P08913 2/20 0.48
ADRA2C P18825 2/20 0.48
SLC6A2 P23975 2/20 0.48
ADRA1A P35348 2/20 0.48
HRH1 P35367 2/20 0.48
HTR2B P41595 2/20 0.48
HTR2A P28223 5/20 0.47
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
UBE2T Q9NPD8 1/20 0.41
ASIC3 Q9UHC3 1/20 0.41
DRD1 P21728 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL7776847 0.91 DRD2 (0.42) DRD2DRD3DRD4HTR7HTR1A
SCHEMBL7773495 0.89 DRD2 (0.48) DRD2DRD3DRD4HTR7HTR1A
SCHEMBL7773460 0.89 DRD2 (0.54) DRD2DRD3DRD4HTR7HTR1A
SCHEMBL7773419 0.89 DRD2 (0.61) DRD2DRD3DRD4HTR7HTR1A
SCHEMBL7856234 0.88 OGA (0.43) DRD2DRD3DRD4HTR7HTR1A
SCHEMBL7773388 0.84 DRD3 (0.51) DRD2DRD3DRD4HTR7HTR1A
Hydrochloric Acid SCHEMBL7775350 0.83 DRD3 (0.50) DRD2DRD3DRD4HTR7HTR1A
SCHEMBL7775417 0.81 DRD2 (0.45) DRD2DRD3DRD4HTR7HTR1A
SCHEMBL7773366 0.81 DRD3 (0.54) DRD2DRD3DRD4HTR7HTR1A
Fumaric Acid SCHEMBL7776886 0.81 DRD2 (0.42) DRD2DRD3DRD4HTR7HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1117663-A2 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 2001-07-25 EP claimed
WO-2000018767-A2 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 2000-04-06 WO claimed
EP-1117663-A2 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 2001-07-25 EP disclosed
WO-2000018767-A2 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 2000-04-06 WO disclosed