SCHEMBL7774160

SCHEMBL7774160

O=C(COc1cccc2ccccc12)N1CCN(c2cc(N3CCCC3)nc(N3CCCC3)n2)CC1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.70
ALDH1A1 P00352 4/20 0.70
MAPT P10636 3/20 0.70
HSD17B10 Q99714 2/20 0.70
TSHR P16473 2/20 0.70
RECQL P46063 1/20 0.70
LMNA P02545 2/20 0.65
HTT P42858 1/20 0.65
NPSR1 Q6W5P4 1/20 0.65
SMN1; SMN2 Q16637 2/20 0.54
MC4R P32245 1/20 0.52
RAB9A P51151 2/20 0.52
GBA1 P04062 3/20 0.52
L3MBTL1 Q9Y468 1/20 0.51
RXFP1 Q9HBX9 1/20 0.51
ADRA1A P35348 2/20 0.51
ADRA1B P35368 2/20 0.51
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
HTR1A P08908 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27979632 0.82 ALDH1A1 (0.82) KDM4EALDH1A1MAPTHSD17B10TSHR
SCHEMBL7769746 0.82 KDM4E (0.69) KDM4EALDH1A1MAPTHSD17B10TSHR
SCHEMBL7776116 0.81 NPC1 (0.70) KDM4EALDH1A1MAPTHSD17B10LMNA
SCHEMBL4379063 0.78 KDM4E (0.82) KDM4EALDH1A1MAPTHSD17B10TSHR
SCHEMBL8906560 0.78 GBA1 (0.65) ALDH1A1LMNAGBA1
SCHEMBL14218031 0.75 ALDH1A1 (0.70) KDM4EALDH1A1MAPTHSD17B10TSHR
SCHEMBL17940608 0.75 ALDH1A1 (0.73) KDM4EALDH1A1MAPTHSD17B10TSHR
SCHEMBL1374171 0.74 ALDH1A1 (0.69) KDM4EALDH1A1MAPTHSD17B10TSHR
SCHEMBL4378942 0.74 KDM4E (0.65) KDM4EALDH1A1MAPTHSD17B10TSHR
SCHEMBL2829296 0.74 KDM4E (0.62) KDM4EALDH1A1MAPTHSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0574906-B1 Piperazine and homopiperazine derivatives, pharmaceutical compositions containing them and process for preparing the same NISSHIN FLOUR MILLING CO (JP) 2001-08-22 EP disclosed
US-5380724-A Inhibitors of lipid peroxidation GYOGYSZERKUTATO INTEZET KFT (HU) 1995-01-10 US disclosed