SCHEMBL7774177

SCHEMBL7774177

COc1cc(C(=O)c2c(N(C)C)sc3cc(OCc4ccccc4)ccc23)ccc1OCC(C)(C)N1CCCC1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ESR1 P03372 11/20 0.39
ESR2 Q92731 11/20 0.39
APP P05067 2/20 0.38
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6595414 0.86 ACHE (0.48) NPC1RAB9AHPGDSMN1; SMN2BCHE
SCHEMBL6171046 0.85 CD274 (0.44) MEN1KMT2AESR1ESR2
SCHEMBL7773957 0.84 ESR1 (0.60) MEN1KMT2AESR1ESR2ACHE
SCHEMBL7447753 0.81 MEN1 (0.44) MEN1KMT2AESR1ESR2
SCHEMBL7414778 0.80 NPC1 (0.41) NPC1RAB9AMEN1KMT2AHPGD
SCHEMBL6171651 0.80 EGFR (0.42) HPGDSMN1; SMN2ESR1ESR2BCHE
SCHEMBL7768225 0.79 TDP1 (0.47) NPC1RAB9AMEN1KMT2AHPGD
SCHEMBL6171041 0.77 ESR1 (0.61) ESR1ESR2
SCHEMBL7774131 0.77 HRH3 (0.43) ESR1ESR2
SCHEMBL6176533 0.77 S1PR1 (0.49) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265575-B1 THROMBIN INHIBITORS ELI LILLY AND COMPANY 2001-07-24 US disclosed
US-6251921-B1 ADMINISTERING THROMBIN INHIBITING DIAMINE COMPOUND TO MAMMAL ELI LILLY AND COMPANY 2001-06-26 US disclosed
US-6025382-A Antithrombotic diamines ELI LILLY AND COMPANY (US) 2000-02-15 US disclosed