SCHEMBL7775495

SCHEMBL7775495

Cc1cccc2[nH]c(C(N)CN3CCN(c4cccc(C(F)(F)F)c4)CC3)nc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.53
ALDH1A1 P00352 4/20 0.53
GAA P10253 4/20 0.53
KDM4E B2RXH2 3/20 0.53
LMNA P02545 1/20 0.53
TP53 P04637 1/20 0.53
GLA P06280 1/20 0.53
ALOX15 P16050 1/20 0.53
ALOX12 P18054 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
MAPK1 P28482 3/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
HTT P42858 1/20 0.48
IGF1R P08069 1/20 0.46
HTR1A P08908 4/20 0.45
POLB P06746 2/20 0.45
GBA1 P04062 1/20 0.45
SMPD1 P17405 1/20 0.45
ABCB11 O95342 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL7775413 0.99 MAPT (0.52) MAPTALDH1A1GAAKDM4ELMNA
SCHEMBL7773489 0.75 MEN1 (0.51) MAPTALDH1A1KDM4ELMNATP53
SCHEMBL7773477 0.75 ALDH1A1 (0.44) MAPTALDH1A1GAAKDM4ELMNA
SCHEMBL11284379 0.74 IGF1R (0.60) MAPTALDH1A1GAAKDM4ELMNA
Bromide SCHEMBL7775425 0.74 MEN1 (0.50) MAPTALDH1A1KDM4ELMNATP53
Bromide SCHEMBL7776842 0.74 ALDH1A1 (0.43) MAPTALDH1A1GAAKDM4ELMNA
SCHEMBL7776872 0.74 DRD4 (0.41) MAPTALDH1A1KDM4EMEN1KMT2A
SCHEMBL7769225 0.74 ADRA1A (0.45) MEN1KMT2AHTR1AADRA1A
Bromide SCHEMBL7773346 0.73 DRD4 (0.41) MAPTALDH1A1KDM4EMEN1KMT2A
Bromide SCHEMBL7773499 0.73 ADRA1A (0.44) MEN1KMT2AHTR1AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1117663-A2 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 2001-07-25 EP claimed
WO-2000018767-A9 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORP (US) 2001-04-19 WO claimed
WO-2000018767-A2 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 2000-04-06 WO claimed