SCHEMBL7777918

SCHEMBL7777918

CCCC(C#N)CC(CC(=O)O)CC(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 2/20 0.36
ADRA1A P35348 2/20 0.36
CACNB3 P54284 1/20 0.36
CACNA1C Q13936 1/20 0.36
PGR P06401 1/20 0.36
HTR2B P41595 1/20 0.36
CACNA2D2 Q9NY47 1/20 0.36
GPR84 Q9NQS5 4/20 0.35
CHRM1 P11229 1/20 0.34
AKR1A1 P14550 1/20 0.34
CHRM3 P20309 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HRH1 P35367 1/20 0.34
DRD3 P35462 1/20 0.34
SLC6A3 Q01959 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
GRIK1 P39086 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26073020 0.84 GPR84 (0.39) ADRA1AGPR84CHRM1AKR1A1CHRM3
SCHEMBL3443498 0.84 GPR84 (0.39) ADRA1AGPR84CHRM1AKR1A1CHRM3
Nitrous Acid SCHEMBL28817705 0.78 GPR84 (0.35) ADRA1AGPR84CHRM1AKR1A1CHRM3
SCHEMBL13339645 0.77 TSHR (0.33)
SCHEMBL4381154 0.76 TSHR (0.34) CACNA2D1ADRA1ACACNB3CACNA1CPGR
SCHEMBL3015727 0.76 TSHR (0.34) CACNA2D1ADRA1ACACNB3CACNA1CPGR
SCHEMBL4387847 0.76 TSHR (0.34) CACNA2D1ADRA1ACACNB3CACNA1CPGR
SCHEMBL29035779 0.76 TSHR (0.34) CACNA2D1ADRA1ACACNB3CACNA1CPGR
SCHEMBL3015730 0.76 TSHR (0.34) CACNA2D1ADRA1ACACNB3CACNA1CPGR
SCHEMBL4378802 0.76 TSHR (0.34) CACNA2D1ADRA1ACACNB3CACNA1CPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1124802-A1 PROCESS FOR PRODUCING 4-ARYLPIPERIDINE-3-CARBINOLS AND RELATED COMPOUNDS Synthon B.V. (NL) 2001-08-22 EP disclosed
WO-2000026187-A1 PROCESS FOR PRODUCING 4-ARYLPIPERIDINE-3-CARBINOLS AND RELATED COMPOUNDS SYNTHON B.V. (NL) 2000-05-11 WO disclosed